SCHEMBL8648668

SCHEMBL8648668

CS(=O)(=O)ONC(=N)NC(=O)/C(=C/c1ccccc1F)c1cccnc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
ATM Q13315 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP1A1 P04798 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP1B1 Q16678 1/20 0.35
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
HIF1A Q16665 1/20 0.34
PTGS2 P35354 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
KMT2A Q03164 2/20 0.34
CAPN1 P07384 1/20 0.34
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
MEN1 O00255 1/20 0.34
PKM P14618 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8650931 0.89 ATM (0.37) ALDH1A1ATMCYP1A2CYP3A4CYP1A1
SCHEMBL8646248 0.89 MAPT (0.43) ALDH1A1ATMCYP1A2CYP3A4CYP1A1
SCHEMBL8647153 0.88 CYP1A1 (0.47) ALDH1A1ATMCYP1A2CYP3A4CYP1A1
SCHEMBL8650932 0.86 NPC1 (0.42) ALDH1A1CYP1A2CYP3A4CYP1A1CYP2D6
SCHEMBL8648666 0.86 ALDH1A1 (0.38) ALDH1A1TDP1ATMCYP1A2CYP3A4
SCHEMBL8644182 0.82 F7 (0.41) ALDH1A1TDP1ATMCYP1A2CYP3A4
SCHEMBL8644322 0.82 MAPT (0.42) ALDH1A1CYP3A4CYP2C19PTGS2SMN1; SMN2
SCHEMBL8646761 0.81 CYP3A4 (0.45) ALDH1A1CYP1A2CYP3A4CYP1A1CYP2D6
SCHEMBL8648674 0.81 KMT2A (0.47) ALDH1A1TDP1CYP3A4CYP2C9CYP2C19
SCHEMBL8643116 0.76 KMT2A (0.37) ALDH1A1ATMSMN1; SMN2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861831-A1 HETEROARYL-SUBSTITUTED ACRYLOYLGUANIDINE DERIVATIVES AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-09-02 EP disclosed