SCHEMBL8648674

SCHEMBL8648674

COc1ccc(/C=C(/C(=O)NC(=N)NOS(C)(=O)=O)c2cccnc2)cc1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.47
MEN1 O00255 1/20 0.47
ALDH1A1 P00352 4/20 0.43
GAA P10253 3/20 0.43
MAPT P10636 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
THRB P10828 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8650932 0.90 NPC1 (0.42) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL8644322 0.89 MAPT (0.42) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL8648671 0.87 KMT2A (0.47) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL8646761 0.87 CYP3A4 (0.45) KMT2AMEN1ALDH1A1MAPTKDM4E
SCHEMBL8643707 0.85 KMT2A (0.50) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL8647153 0.84 CYP1A1 (0.47) KMT2AMEN1ALDH1A1GAAMAPT
SCHEMBL8650931 0.82 ATM (0.37) ALDH1A1GAAMAPTKDM4ELMNA
SCHEMBL8648668 0.81 ALDH1A1 (0.35) KMT2AMEN1ALDH1A1MAPTTDP1
SCHEMBL8646248 0.81 MAPT (0.43) KMT2AMEN1ALDH1A1MAPTKDM4E
SCHEMBL8647072 0.79 ALDH1A1 (0.52) KMT2AMEN1ALDH1A1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0861831-A1 HETEROARYL-SUBSTITUTED ACRYLOYLGUANIDINE DERIVATIVES AND MEDICINAL COMPOSITION THEREOF YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1998-09-02 EP disclosed