SCHEMBL8649188

SCHEMBL8649188

Cc1ccc(S(=O)(=O)OCCCc2coc3ccc(Cl)cc23)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 3/20 0.40
THRB P10828 2/20 0.39
TP53 P04637 2/20 0.38
CA12 O43570 4/20 0.38
CA1 P00915 4/20 0.38
CA9 Q16790 4/20 0.38
MTNR1A P48039 3/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HSD17B10 Q99714 1/20 0.36
CA2 P00918 3/20 0.36
PSMD10 O75832 1/20 0.36
FBP1 P09467 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 2/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8649142 0.93 PDE10A (0.41) PDE10ATHRBTP53CA12CA1
SCHEMBL8650318 0.87 THRB (0.39) PDE10ATHRBCA12CA1CA9
SCHEMBL8649534 0.86 MTNR1A (0.55) CA12CA1CA9MTNR1AMAPT
SCHEMBL8647162 0.84 CA2 (0.44) CA12CA1CA9CA2PSMD10
SCHEMBL8788431 0.80 CYP1A2 (0.43) PDE10ATHRBTP53CA12CA1
SCHEMBL9215791 0.78 SLC6A4 (0.52) TP53MTNR1AHSD17B10KMT2AMAPT
SCHEMBL8787860 0.77 CYP1A2 (0.45) PDE10ATHRBTP53CA12CA1
SCHEMBL8648707 0.76 CA2 (0.46) CA12CA1CA9CA2KMT2A
SCHEMBL16432776 0.75 SLC6A4 (0.51) TP53MTNR1AHSD17B10KMT2AMAPT
SCHEMBL7723972 0.74 CNR2 (0.54) THRBALDH1A1PSMD10KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763444-A CENTRAL NERVOUS SYSTEM AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-06-09 US disclosed
EP-0761666-A2 Antidepressant 1-arylalkyl-4-(alkoxypyridinyl)- or 4-(alkoxypyrimidinyl)piperazine derivatives BRISTOL-MYERS SQUIBB COMPANY (US) 1997-03-12 EP disclosed