SCHEMBL8650318

SCHEMBL8650318

Cc1ccc(S(=O)(=O)OCCCc2coc3ccc(F)cc23)cc1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.39
CA12 O43570 4/20 0.38
CA1 P00915 4/20 0.38
CA9 Q16790 4/20 0.38
MTNR1A P48039 3/20 0.38
PDE10A Q9Y233 3/20 0.37
HTR1A P08908 2/20 0.37
CA2 P00918 3/20 0.36
PSMD10 O75832 1/20 0.36
POLB P06746 1/20 0.35
MAPT P10636 1/20 0.35
HTR6 P50406 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8649188 0.87 PDE10A (0.40) THRBCA12CA1CA9MTNR1A
SCHEMBL8649534 0.86 MTNR1A (0.55) CA12CA1CA9MTNR1APOLB
SCHEMBL8647162 0.84 CA2 (0.44) CA12CA1CA9CA2PSMD10
SCHEMBL8788242 0.80 THRB (0.41) THRBCA12CA1CA9MTNR1A
SCHEMBL8649142 0.80 PDE10A (0.41) THRBCA12CA1CA9MTNR1A
SCHEMBL8650329 0.78 MTNR1A (0.46) THRBCA12CA1CA9MTNR1A
SCHEMBL4351623 0.78 MPO (0.54) HTR1A
SCHEMBL8648707 0.76 CA2 (0.46) CA12CA1CA9CA2
SCHEMBL7813034 0.76 MTNR1A (0.46) MTNR1APDE10AHTR1AHTR6
SCHEMBL9213281 0.76 HTR2A (0.48) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763444-A CENTRAL NERVOUS SYSTEM AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-06-09 US disclosed
EP-0761666-A2 Antidepressant 1-arylalkyl-4-(alkoxypyridinyl)- or 4-(alkoxypyrimidinyl)piperazine derivatives BRISTOL-MYERS SQUIBB COMPANY (US) 1997-03-12 EP disclosed