SCHEMBL8649495

SCHEMBL8649495

CC(C)(OS(=O)(=O)C(F)(F)F)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
TSHR P16473 1/20 0.33
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
PPARA Q07869 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1784844 0.77 ALDH1A1 (0.34) ALDH1A1L3MBTL1TSHR
SCHEMBL1784841 0.77 ALDH1A1 (0.34) ALDH1A1L3MBTL1TSHR
SCHEMBL2335624 0.75 TSHR (0.36) ALDH1A1TSHRMEN1CYP1A2CYP3A4
SCHEMBL700952 0.74 ADORA3 (0.33) ALDH1A1L3MBTL1PPARA
SCHEMBL700953 0.74 ADORA3 (0.33) ALDH1A1L3MBTL1PPARA
SCHEMBL701748 0.74 ADORA3 (0.33) ALDH1A1L3MBTL1PPARA
SCHEMBL145452 0.74 CA1 (0.33)
SCHEMBL30655945 0.74 CA1 (0.33)
SCHEMBL776698 0.74 CA1 (0.33)
SCHEMBL14669110 0.74 CA1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5847135-A Inhibitors of interleukin-1β converting enzyme VERTEX PHARMACEUTICALS, INCORPORATED (US) 1998-12-08 US disclosed
EP-0784628-A1 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME Vertex Pharmaceuticals Incorporated (US) 1997-07-23 EP disclosed
WO-1995035308-A1 INHIBITORS OF INTERLEUKIN-1β CONVERTING ENZYME VERTEX PHARMACEUTICALS INCORPORATED (US) 1995-12-28 WO disclosed