SCHEMBL8655703

SCHEMBL8655703

O=C1c2c(oc(-c3ccc(O)cc3)c2CCCCCCN2CCCCC2)C=CC1O

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 10/20 0.43
ESR2 Q92731 7/20 0.43
CYP2D6 P10635 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
KCNH2 Q12809 2/20 0.34
HRH1 P35367 1/20 0.33
XDH P47989 1/20 0.33
BCL9 O00512 2/20 0.33
CTNNB1 P35222 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8654623 0.78 ESR1 (0.44) ESR1ESR2CYP2D6SIGMAR1KCNH2
SCHEMBL8653155 0.78 ESR1 (0.39) ESR1ESR2CYP2D6
SCHEMBL8636932 0.71 ESR1 (0.51) ESR1ESR2KCNH2XDH
SCHEMBL8637238 0.71 XDH (0.49) ESR1ESR2CYP2D6XDH
SCHEMBL7647862 0.63 ESR1 (0.61) ESR1ESR2SIGMAR1HRH1
SCHEMBL8641220 0.61 ESR1 (0.62) ESR1ESR2CYP2D6SIGMAR1KCNH2
SCHEMBL9027633 0.59 ESR1 (0.43) ESR1ESR2SIGMAR1KCNH2HRH1
SCHEMBL8196023 0.58 ESR1 (0.44) ESR1ESR2CYP2D6SIGMAR1KCNH2
SCHEMBL8654530 0.58 PTPN1 (0.37) ESR1ESR2
SCHEMBL7367096 0.57 HRH3 (0.72) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0516257-B1 Phenylbenzo[b]furans and -thiophenes, procedures for their preparation, and pharmaceutical compositions containing the same SCHERING AG (DE) 1998-08-05 EP claimed