SCHEMBL8655825

SCHEMBL8655825

FC(F)(F)c1ccc(Oc2ccc(COc3c(Cl)cc(OCC=C(Cl)Cl)cc3Cl)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 10/20 0.41
PPARD Q03181 2/20 0.40
PPARA Q07869 2/20 0.40
PPARG P37231 2/20 0.39
THRB P10828 1/20 0.39
MAOA P21397 3/20 0.38
FFAR1 O14842 2/20 0.38
ALOX5 P09917 1/20 0.38
PSEN1 P49768 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8408840 0.95 MAOB (0.42) MAOBPPARDPPARAPPARGMAOA
SCHEMBL8655830 0.86 FFAR1 (0.42) PPARGTHRBFFAR1
SCHEMBL8405935 0.85 GCGR (0.40) MAOBFFAR1
SCHEMBL8407176 0.84 MRGPRX4 (0.42) PPARDTHRB
SCHEMBL8658648 0.84 PTGES (0.37) MAOBPPARDPPARAPPARGTHRB
SCHEMBL8655774 0.83 RXRA (0.42) MAOB
SCHEMBL8405312 0.83 MAOB (0.49) MAOBPPARDPPARATHRBMAOA
SCHEMBL8407561 0.83 MAOB (0.47) MAOBTHRBFFAR1
SCHEMBL8659996 0.83 FFAR1 (0.36) MAOBPPARDPPARAPPARGTHRB
SCHEMBL8405597 0.82 MAOB (0.39) MAOBPPARDPPARATHRBFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0722430-B1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL CO (JP) 1998-10-21 EP disclosed
EP-0722430-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1996-07-24 EP disclosed
WO-1996004228-A1 DIHALOPROPENE COMPOUNDS, INSECTICIDAL/ACARICIDAL AGENTS CONTAINING SAME, AND INTERMEDIATES FOR THEIR PRODUCTION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1996-02-15 WO disclosed