SCHEMBL8656643

SCHEMBL8656643

CCN(c1ccc(C(C)(C)N)cc1)S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.54
NFE2L2 Q16236 1/20 0.54
CNR2 P34972 3/20 0.54
LMNA P02545 3/20 0.52
CNR1 P21554 2/20 0.52
MAPT P10636 2/20 0.52
ESR1 P03372 2/20 0.51
ALDH1A1 P00352 3/20 0.50
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
CYP2C19 P33261 1/20 0.49
NPSR1 Q6W5P4 2/20 0.49
NR3C1 P04150 1/20 0.49
PGR P06401 1/20 0.49
HSD11B1 P28845 1/20 0.49
NR1I2 O75469 1/20 0.47
RORA P35398 1/20 0.47
RORC P51449 1/20 0.47
NR1H2 P55055 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5622498 0.87 KEAP1 (0.68) KEAP1NFE2L2CNR2LMNACNR1
SCHEMBL8656600 0.84 HCRTR2 (0.52) LMNAMAPTESR1ALDH1A1NPSR1
SCHEMBL7182031 0.81 ESR1 (0.79) KEAP1NFE2L2CNR2LMNACNR1
SCHEMBL8657231 0.81 RORC (0.53) MAPTESR1TSHRNPSR1NR3C1
SCHEMBL28728523 0.80 CNR1 (0.70) KEAP1NFE2L2CNR2LMNACNR1
SCHEMBL1039041 0.76 HCRTR2 (0.77) KEAP1NFE2L2MAPTALDH1A1TP53
SCHEMBL5622632 0.76 KEAP1 (0.64) KEAP1NFE2L2CNR2LMNACNR1
SCHEMBL1630208 0.73 KEAP1 (0.81) KEAP1NFE2L2MAPT
SCHEMBL5622935 0.73 KEAP1 (0.61) KEAP1NFE2L2CNR2LMNACNR1
SCHEMBL5624485 0.73 KEAP1 (0.61) KEAP1NFE2L2CNR2LMNACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780642-A NON-STEROIDAL ANTIINFLAMMATORY AGENT WHICH BLOCKS RELEASE OF ARACHIDONIC ACID FROM PHOSPHOLIPIDS; SIDE EFFECT REDUCTION KNOLL AKTIENGESELLSCHAFT (DE) 1998-07-14 US disclosed