SCHEMBL8657231

SCHEMBL8657231

CCN(c1ccc(C(C)(C)N)cc1)S(=O)(=O)c1ccc(C#N)cc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RORC P51449 7/20 0.53
NR1I2 O75469 2/20 0.53
RORA P35398 2/20 0.53
NR1H2 P55055 2/20 0.53
RORB Q92753 2/20 0.53
NR1H4 Q96RI1 2/20 0.53
HCRTR2 O43614 2/20 0.53
ESR1 P03372 2/20 0.50
HSD11B1 P28845 1/20 0.48
NR1H3 Q13133 2/20 0.47
NR3C1 P04150 1/20 0.46
PGR P06401 1/20 0.46
TSHR P16473 1/20 0.44
MAPK1 P28482 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
KDM1A O60341 2/20 0.43
NPSR1 Q6W5P4 2/20 0.42
MAPT P10636 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6828511 0.82 HCRTR2 (0.73) RORCHCRTR2ESR1KDM1A
SCHEMBL8656643 0.81 KEAP1 (0.54) RORCNR1I2RORANR1H2RORB
SCHEMBL8656600 0.75 HCRTR2 (0.52) HCRTR2ESR1KMT2ANPSR1MAPT
SCHEMBL156260 0.73 KIF11 (0.59) TSHR
SCHEMBL28383987 0.72 HCRTR2 (0.46) RORCNR1I2RORANR1H2RORB
SCHEMBL30326344 0.72 HCRTR2 (0.46) RORCNR1I2RORANR1H2RORB
SCHEMBL3636387 0.71 LMNA (0.63) HCRTR2KMT2AKDM1AMAPT
SCHEMBL21339855 0.70 CYP19A1 (0.51) RORCNR1I2RORANR1H2RORB
SCHEMBL15853614 0.69 HSD11B1 (0.76) RORCNR1I2RORANR1H2RORB
SCHEMBL14350007 0.68 RORC (0.54) RORCNR1I2RORANR1H2RORB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780642-A NON-STEROIDAL ANTIINFLAMMATORY AGENT WHICH BLOCKS RELEASE OF ARACHIDONIC ACID FROM PHOSPHOLIPIDS; SIDE EFFECT REDUCTION KNOLL AKTIENGESELLSCHAFT (DE) 1998-07-14 US disclosed