SCHEMBL8659490

SCHEMBL8659490

Fc1cc2[nH]c(SCc3ccc(Cl)c(Cl)c3)nc2cc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRL1 P41146 9/20 0.49
DAO P14920 1/20 0.48
TXN P10599 1/20 0.47
RAB9A P51151 3/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
PRKAG1 P54619 2/20 0.47
PRKAA2 P54646 2/20 0.47
PRKAB1 Q9Y478 2/20 0.47
NPC1 O15118 2/20 0.47
LMNA P02545 1/20 0.47
HTT P42858 1/20 0.47
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2E1 P05181 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C8 P10632 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2B6 P20813 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALOX5 P09917 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL211295 0.82 ALOX5 (0.67) OPRL1SMN1; SMN2PRKAG1PRKAA2PRKAB1
SCHEMBL12963079 0.81 OPRL1 (0.60) OPRL1RAB9ASMN1; SMN2NPC1LMNA
SCHEMBL8631022 0.80 RAB9A (0.67) RAB9ASMN1; SMN2NPC1LMNAHTT
SCHEMBL8291911 0.78 SMN1; SMN2 (0.46) OPRL1RAB9ASMN1; SMN2PRKAG1PRKAA2
SCHEMBL8291917 0.77 ALOX5 (0.64) OPRL1SMN1; SMN2PRKAG1PRKAA2PRKAB1
SCHEMBL9692985 0.77 RAB9A (0.60) DAORAB9ASMN1; SMN2NPC1LMNA
SCHEMBL4207157 0.76 RAB9A (0.58) RAB9ASMN1; SMN2PRKAG1PRKAA2PRKAB1
SCHEMBL12963220 0.76 CYP1A2 (0.52) OPRL1TXNRAB9ASMN1; SMN2PRKAG1
SCHEMBL8634298 0.75 MAPT (0.61) DAORAB9ASMN1; SMN2NPC1LMNA
SCHEMBL12932936 0.75 CYP1A2 (0.53) OPRL1TXNSMN1; SMN2PRKAG1PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0830346-A1 2-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PRODUCTS CORPORATION (US) 1998-03-25 EP claimed
US-5684030-A HYPOTENSIVE AGENTS, ANTIPROLIFERATION AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1997-11-04 US claimed
WO-1996040645-A1 2-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PRODUCTS CORPORATION (US) 1996-12-19 WO claimed
EP-0830346-A1 2-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PRODUCTS CORPORATION (US) 1998-03-25 EP disclosed
US-5684030-A HYPOTENSIVE AGENTS, ANTIPROLIFERATION AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1997-11-04 US disclosed
WO-1996040645-A1 2-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF SMOOTH MUSCLE CELL PROLIFERATION AMERICAN HOME PRODUCTS CORPORATION (US) 1996-12-19 WO disclosed