SCHEMBL8660177

SCHEMBL8660177

COc1ccc(-c2cc3c(cc2-c2ccccc2S(N)(=O)=O)OCO3)cc1OC

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.47
TOP2A P11388 1/20 0.45
PTGS1 P23219 4/20 0.44
BRD4 O60885 1/20 0.42
P2RX3 P56373 3/20 0.42
USP2 O75604 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
MAPT P10636 1/20 0.41
KIT P10721 1/20 0.41
F10 P00742 3/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
CYP19A1 P11511 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8662796 0.91 POLB (0.41) PTGS2TOP2APTGS1BRD4P2RX3
SCHEMBL8659929 0.90 PTGS2 (0.58) PTGS2PTGS1BRD4P2RX3MAPT
SCHEMBL8656219 0.90 PTGS2 (0.46) PTGS2PTGS1F10
SCHEMBL8661650 0.90 PTGS2 (0.46) PTGS2PTGS1BRD4P2RX3MAPT
SCHEMBL8656787 0.88 PTGS2 (0.39) PTGS2TOP2APTGS1P2RX3USP2
SCHEMBL8657255 0.88 CA9 (0.44) PTGS2PTGS1BRD4MAPTF10
SCHEMBL8661261 0.87 PTGS1 (0.40) PTGS2PTGS1P2RX3ALDH1A1HSP90AA1
SCHEMBL8660155 0.87 PTGS2 (0.40) PTGS2PTGS1P2RX3ALDH1A1HSP90AA1
SCHEMBL8658302 0.87 PTGS2 (0.39) PTGS2PTGS1BRD4P2RX3F10
SCHEMBL8661927 0.84 PTGS2 (0.36) PTGS2PTGS1P2RX3ALDH1A1HSP90AA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739166-A ALKYLSULFONYL OR AMINOSULFONYL SUBSTITUTED AROMATIC COMPOUNDS AS NON-STEROIDAL ANTIINFLAMMATORY AGENT G.D. SEARLE & CO. (US) 1998-04-14 US disclosed