SCHEMBL8660425

SCHEMBL8660425

Cc1nn(-c2ccccc2)c(=O)n1C(F)F

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.47
PPOX P50336 1/20 0.43
ADORA3 P0DMS8 3/20 0.42
HIF1A Q16665 1/20 0.42
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
HTT P42858 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CA9 Q16790 1/20 0.39
MAPK1 P28482 2/20 0.39
NTRK1 P04629 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7067774 0.84 PPOX (0.47) ROCK2PPOXADORA3CA9
SCHEMBL9427767 0.82 PPOX (0.44) PPOXADORA3ADORA2AADORA1ALDH1A1
SCHEMBL6659733 0.80 PPOX (0.46) PPOXALDH1A1
SCHEMBL9427869 0.79 ABHD16A (0.50) HTTALDH1A1
SCHEMBL9120418 0.78 PPOX (0.57) PPOXALDH1A1
SCHEMBL29575373 0.77 PPOX (0.45) ROCK2PPOXADORA3LMNA
SCHEMBL29575134 0.76 PPOX (0.55) PPOXHTTALDH1A1
SCHEMBL7658153 0.75 ADORA3 (0.51) ADORA3HIF1AADORA2AADORA1ALDH1A1
SCHEMBL9428146 0.74 PPOX (0.45) PPOX
SCHEMBL10562068 0.74 ROCK2 (0.47) ROCK2PPOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8669371-B2 Regioselective chlorination of the phenyl ring of 4,5-dihydro-1-phenyl-1H-1,2,4-triazol-5-ones TAGROS CHEMICALS INDIA PVT LTD (IN) 2014-03-11 US claimed
US-20130072689-A1 Regioselective chlorination of the phenyl ring of 4,5-dihydro-1-phenyl-1H-1,2,4-triazol-5-ones TAGROS CHEMICALS INDIA, LTD. (IN) 2013-03-21 US claimed
US-5468868-A Process for the selective chlorination of 4,5-dihydro-1-phenyl-1H-1,2,4-triazol-5-one FMC CORPORATION (US) 1995-11-21 US claimed
CN-111689915-A Preparation method of 1- (2, 4-dichlorophenyl) -4-difluoromethyl-3-methyl-1H-1, 2, 4-triazole-5-ketone 湖南斯派克科技股份有限公司 2020-09-22 CN disclosed
US-8669371-B2 Regioselective chlorination of the phenyl ring of 4,5-dihydro-1-phenyl-1H-1,2,4-triazol-5-ones TAGROS CHEMICALS INDIA PVT LTD (IN) 2014-03-11 US disclosed
US-20130072689-A1 Regioselective chlorination of the phenyl ring of 4,5-dihydro-1-phenyl-1H-1,2,4-triazol-5-ones TAGROS CHEMICALS INDIA, LTD. (IN) 2013-03-21 US disclosed
US-5756755-A Difluoromethylation of 4,5-dihydro-1-phenyl-3-methyl-1,2,4-triazol-5(1H)-ones with glymes as solvents FMC CORPORATION (US) 1998-05-26 US disclosed
WO-1997003972-A1 DIFLUOROMETHYLATION OF A PHENYL TRIAZOLINONE FMC CORPORATION (US) 1997-02-06 WO disclosed
US-5468868-A Process for the selective chlorination of 4,5-dihydro-1-phenyl-1H-1,2,4-triazol-5-one FMC CORPORATION (US) 1995-11-21 US disclosed
US-5438149-A Reacting with chlorodifluoromethane and potassium carbonate while heating in solvent of dimethylformamide, 1-methyl-2-pyrrolidone or N,N-dimethylacetamide FMC CORPORATION (US) 1995-08-01 US disclosed