SCHEMBL8660847

SCHEMBL8660847

COC(=O)c1c(O)ccc2ocnc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.49
CA1 P00915 4/20 0.49
CA2 P00918 4/20 0.49
CA7 P43166 4/20 0.49
CA9 Q16790 4/20 0.49
CA14 Q9ULX7 4/20 0.49
KDM4E B2RXH2 3/20 0.40
HSD17B10 Q99714 2/20 0.40
XDH P47989 1/20 0.38
PIN1 Q13526 1/20 0.36
CYP3A4 P08684 2/20 0.36
ACHE P22303 1/20 0.36
LCK P06239 1/20 0.35
LMNA P02545 4/20 0.35
TSHR P16473 2/20 0.35
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
HPGD P15428 3/20 0.34
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8674319 0.75 CA12 (0.49) CA12CA1CA2CA7CA9
SCHEMBL29704385 0.73 TOP2A (0.47) KDM4EHSD17B10PIN1LMNATSHR
SCHEMBL19644298 0.73 TOP2A (0.47) KDM4EHSD17B10PIN1LMNATSHR
SCHEMBL160098 0.73 CA12 (0.77) CA12CA1CA2CA7CA9
SCHEMBL8655395 0.73 ALDH1A1 (0.45) CYP3A4ALDH1A1SMN1; SMN2
SCHEMBL27033003 0.71 CA12 (0.52) CA12CA1CA2CA7CA9
SCHEMBL27033243 0.70 FGFR1 (0.33) KDM4EHSD17B10XDHLMNAMTNR1A
SCHEMBL8980290 0.69 PIN1 (0.39) CA1CA2KDM4EHSD17B10XDH
SCHEMBL28508446 0.69 PIN1 (0.50) CA1CA2CA9KDM4EHSD17B10
SCHEMBL161350 0.68 CA12 (0.68) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770544-A TRIAZINES KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1998-06-23 US disclosed
US-5616537-A Condensed heterocyclic derivatives and herbicides KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1997-04-01 US disclosed
EP-0606489-A1 CONDENSED HETEROCYCLIC DERIVATIVE AND WEEDKILLER KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1994-07-20 EP disclosed