SCHEMBL8664405

SCHEMBL8664405

Nc1ccc(C(=O)N(CCN2CCC(C(=O)c3ccccc3)CC2)c2cccnc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 6/20 0.50
HTR2A P28223 1/20 0.46
CHRM3 P20309 1/20 0.45
ACHE P22303 2/20 0.43
KCNH2 Q12809 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8716555 0.96 PTGIR (0.46) PTGIRHTR2ACHRM3ACHEKCNH2
Maleic Acid SCHEMBL8716551 0.96 PTGIR (0.46) PTGIRHTR2ACHRM3ACHEKCNH2
SCHEMBL8710951 0.93 SLC18A3 (0.50) HTR2AACHE
SCHEMBL8710974 0.87 PTGIR (0.47) PTGIRHTR2ACHRM3ACHEKCNH2
SCHEMBL8711151 0.87 HTR2A (0.57) PTGIRHTR2ACHRM3ACHEKCNH2
SCHEMBL8710869 0.84 ACHE (0.56) PTGIRHTR2AACHE
SCHEMBL8711207 0.84 LMNA (0.49) HTR2A
Fumaric Acid SCHEMBL8711104 0.84 PTGIR (0.44) PTGIRHTR2ACHRM3ACHE
Fumaric Acid SCHEMBL8711107 0.84 PTGIR (0.44) PTGIRHTR2ACHRM3ACHE
SCHEMBL8711319 0.83 SLC18A3 (0.49) HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-10077271-A None JP disclosed
JP-H1077271-A CIRCULATORY ORGAN MEDICINE CONTAINING 3-PYRIDYLAMINO COMPOUND OR ITS SALT TOA EIYOO KK 1998-03-24 JP disclosed
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed