SCHEMBL8711151

SCHEMBL8711151

O=C(c1ccccc1)C1CCN(CCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2cccnc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.57
ACHE P22303 2/20 0.53
PTGIR P43119 3/20 0.47
CHRM3 P20309 2/20 0.47
CHRM2 P08172 1/20 0.47
SLC18A3 Q16572 1/20 0.45
ALDH1A1 P00352 3/20 0.43
MAPT P10636 1/20 0.43
HSD11B1 P28845 1/20 0.41
MGLL Q99685 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710852 0.93 HSD11B1 (0.51) HTR2AACHESLC18A3HSD11B1
SCHEMBL8664405 0.87 PTGIR (0.50) HTR2AACHEPTGIRCHRM3KCNH2
SCHEMBL8715718 0.85 HTR2A (0.61) HTR2AACHEPTGIRCHRM3CHRM2
SCHEMBL8710974 0.84 PTGIR (0.47) HTR2AACHEPTGIRCHRM3MAPT
Maleic Acid SCHEMBL8716551 0.83 PTGIR (0.46) HTR2AACHEPTGIRCHRM3KCNH2
Fumaric Acid SCHEMBL8716555 0.83 PTGIR (0.46) HTR2AACHEPTGIRCHRM3KCNH2
SCHEMBL9232680 0.81 HSD11B1 (0.56) HTR2AACHEHSD11B1MGLL
Fumaric Acid SCHEMBL8711107 0.81 PTGIR (0.44) HTR2AACHEPTGIRCHRM3MAPT
SCHEMBL8711207 0.81 LMNA (0.49) HTR2ASLC18A3
Fumaric Acid SCHEMBL8711104 0.81 PTGIR (0.44) HTR2AACHEPTGIRCHRM3MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed