SCHEMBL8667012

SCHEMBL8667012

CCN(C)c1c(Nc2cccnc2)c(=O)c1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD52 P43351 1/20 0.41
KMT2A Q03164 1/20 0.41
ADAMTS5 Q9UNA0 1/20 0.41
TDP2 O95551 1/20 0.41
NSD2 O96028 1/20 0.41
CXCR2 P25025 1/20 0.40
NOTUM Q6P988 1/20 0.40
CHRNB2 P17787 2/20 0.39
CHRNA4 P43681 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ADRA2A P08913 2/20 0.38
ADRA2B P18089 2/20 0.38
ADRA2C P18825 2/20 0.38
ITGB1 P05556 1/20 0.38
ITGA4 P13612 1/20 0.38
TDO2 P48775 1/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37
TRPV1 Q8NER1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7351783 0.85 RAD52 (0.45) RAD52KMT2ATDP2NSD2CXCR2
SCHEMBL7350556 0.74 MAPKAPK2 (0.43) RAD52KMT2ATDP2NSD2LMNA
SCHEMBL19956891 0.74 KMT2A (0.49) RAD52KMT2ATDP2NSD2ADRA2A
SCHEMBL4023982 0.73 POLB (0.55) RAD52KMT2ASMN1; SMN2KDM4ELMNA
SCHEMBL7346763 0.71 TDO2 (0.50) RAD52KMT2ATDP2NSD2ADRA2A
SCHEMBL10082731 0.71 CXCR2 (0.54) KMT2AADAMTS5CXCR2ITGB1ITGA4
SCHEMBL2771874 0.71 POLB (0.46) RAD52KMT2ATDP2NSD2KDM4E
SCHEMBL7349452 0.71 PLK1 (0.55) RAD52KMT2ATDP2NSD2
SCHEMBL15061601 0.68 LMNA (0.54) KMT2ANOTUMSMN1; SMN2KDM4ELMNA
SCHEMBL6987237 0.68 KMT2A (0.42) RAD52KMT2ATDP2NSD2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0729457-B1 DIAMINOCYCLOBUTENE-3,4-DIONES AS SMOOTH MUSCLE RELAXANTS AMERICAN HOME PROD (US) 1998-12-23 EP claimed