Aspartic Acid

Aspartic Acid

SCHEMBL8667052

Cc1ccc(S(=O)(=O)NCC(=O)O)cc1.N[C@@H](CC(=O)O)C(=O)O

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

SSTR1SSTR2SSTR3SSTR5

The experimentally established mechanism targets of Aspartic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 2/20 0.51
GBA1 P04062 1/20 0.51
GAA P10253 1/20 0.51
MMP12 P39900 1/20 0.51
SLC1A3 P43003 1/20 0.50
SLC1A2 P43004 1/20 0.50
SLC1A1 P43005 1/20 0.50
MMP2 P08253 1/20 0.49
MMP3 P08254 1/20 0.49
MMP7 P09237 1/20 0.49
MMP9 P14780 1/20 0.49
MMP13 P45452 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.47
ALDH1A1 P00352 2/20 0.46
KMT2A Q03164 1/20 0.46
APEX1 P27695 1/20 0.46
CA12 O43570 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
ATM Q13315 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL760439 0.85 MMP1 (0.67) MMP1GAAMMP12MMP2MMP3
Aspartic Acid SCHEMBL10590014 0.81 KDM4E (0.47) SLC1A3SLC1A2SLC1A1SMN1; SMN2ALDH1A1
Aspartic Acid SCHEMBL10590016 0.81 KDM4E (0.47) SLC1A3SLC1A2SLC1A1SMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL6739604 0.80 GBA1 (0.65) MMP1GBA1SLC1A3SLC1A2SLC1A1
Hydrochloric Acid SCHEMBL6739598 0.80 GBA1 (0.65) MMP1GBA1SLC1A3SLC1A2SLC1A1
SCHEMBL1664363 0.79 LARS1 (0.59) MMP1GBA1GAASLC1A3SLC1A2
SCHEMBL8023841 0.79 GBA1 (0.55) GBA1SLC1A3SLC1A2SLC1A1ALDH1A1
SCHEMBL7329249 0.79 GBA1 (0.63) GBA1SLC1A3SLC1A2SLC1A1ALDH1A1
Hydrochloric Acid SCHEMBL8567005 0.78 GBA1 (0.54) GBA1SLC1A3SLC1A2SLC1A1ALDH1A1
SCHEMBL8451097 0.77 MMP9 (0.57) MMP1GAAMMP12MMP2MMP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691986-B1 NOVEL PROCESSES AND INTERMEDIATE COMPOUNDS FOR THE PREPARATION OF PLATELET CLYCOPROTEIN IIb/IIIa INHIBITORS DU PONT MERCK PHARMA (US) 1998-12-02 EP disclosed
US-5817749-A CYCLIC PENTAPEPTIDES DUPONT PHARMACEUTICALS COMPANY (US) 1998-10-06 US disclosed
EP-0691986-A1 NOVEL PROCESSES AND INTERMEDIATE COMPOUNDS FOR THE PREPARATION OF PLATELET CLYCOPROTEIN IIb/IIIa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-01-17 EP disclosed
WO-1994022909-A1 NOVEL PROCESSES AND INTERMEDIATE COMPOUNDS FOR THE PREPARATION OF PLATELET CLYCOPROTEIN IIb/IIIa INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1994-10-13 WO disclosed