SCHEMBL8668191

SCHEMBL8668191

COC(=O)C(OC)c1ccc(OC2CCN(C(C)=O)CC2)cc1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
F10 P00742 5/20 0.50
PRSS1 P07477 5/20 0.50
PRSS2 P07478 5/20 0.50
PRSS3 P35030 5/20 0.50
PLG P00747 4/20 0.49
SRD5A1 P18405 1/20 0.46
NAMPT P43490 1/20 0.46
ACACB O00763 7/20 0.45
CYP4F2 P78329 1/20 0.44
CYP4A11 Q02928 1/20 0.44
HRH3 Q9Y5N1 1/20 0.43
F2 P00734 2/20 0.43
RORC P51449 1/20 0.43
EPHX2 P34913 1/20 0.42
CHEK2 O96017 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664984 0.89 F10 (0.58) F10PRSS1PRSS2PRSS3PLG
SCHEMBL7364906 0.85 GPR119 (0.59) HRH3CHEK2
SCHEMBL18672909 0.81 MEN1 (0.56) F10PRSS1PRSS2PRSS3PLG
SCHEMBL9013886 0.77 CASP6 (0.53) F10PRSS1PRSS2PRSS3PLG
SCHEMBL16220677 0.77 EPHX2 (0.56) NAMPTCYP4F2CYP4A11HRH3RORC
SCHEMBL24596887 0.76 CYP4F2 (0.51) F10PRSS1PRSS2PRSS3SRD5A1
SCHEMBL2096831 0.76 EPHX2 (0.55) NAMPTACACBCYP4F2CYP4A11EPHX2
Hydrochloric Acid SCHEMBL9014030 0.76 CASP6 (0.51) F10PRSS1PRSS2PRSS3PLG
SCHEMBL31370640 0.76 ALDH1A1 (0.55) SRD5A1NAMPTCYP4F2CYP4A11HRH3
SCHEMBL2091338 0.75 EPHX2 (0.57) SRD5A1NAMPTCYP4F2CYP4A11RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756504-A TREATMENT OF DYSMENORRHEA, PREVENTION OF PREMATURE LABOR MERCK & CO., INC. (US) 1998-05-26 US disclosed
US-5464788-A Stopping labor MERCK & CO., INC. (US) 1995-11-07 US disclosed
WO-1995025443-A1 TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 1995-09-28 WO disclosed