SCHEMBL8668672

SCHEMBL8668672

CCc1ncnc(N)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.36
HEXA P06865 2/20 0.36
HEXB P07686 2/20 0.36
MEN1 O00255 1/20 0.36
SLC22A1 O15245 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
HTR2A P28223 1/20 0.36
ADRA1A P35348 1/20 0.36
HTR2B P41595 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KMT2A Q03164 1/20 0.36
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13064098 0.84 SELE (0.35) SELEVCAM1
SCHEMBL16712847 0.78 RPS6KB1 (0.30) RPS6KB1
SCHEMBL28518966 0.78 AHCY (0.33) ADORA2AADORA1ADORA2B
SCHEMBL3641399 0.77 SELE (0.40) ALDH1A1LMNAPDE4DSMN1; SMN2SELE
SCHEMBL30828905 0.76 SELE (0.32) SELEVCAM1
SCHEMBL16712851 0.76 SELE (0.32) SELEVCAM1
SCHEMBL12323407 0.76 NOS2 (0.45) DHFRADORA2AADORA1PI4KAPI4K2B
SCHEMBL8718664 0.76 SELE (0.32) SELEVCAM1
SCHEMBL15155111 0.75 RPS6KB1 (0.32) RPS6KB1
SCHEMBL8491244 0.74 SELE (0.31) SELEVCAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3702355-B1 SUBSTITUTED PYRAZOLE COMPOUNDS CONTAINING PYRIMIDINE, THE PREPARATION AND APPLICATION THEREOF SHENYANG SINOCHEM AGROCHEMICALS R & D CO LTD (CN) 2022-01-12 EP disclosed
EP-2913325-B1 SUBSTITUTED PYRIMIDINE COMPOUND AND USES THEREOF SHENYANG SINOCHEM AGROCHEMICALS R & D CO LTD (CN) 2021-04-21 EP disclosed
EP-3299366-B1 SUBSTITUTED PYRAZOLE COMPOUNDS CONTAINING PYRIMIDINE AND PREPARATION METHOD AND USE THEREOF AS PESTICIDES SHENYANG SINOCHEM AGROCHEMICALS R & D CO LTD (CN) 2020-09-09 EP disclosed
EP-3702355-A1 SUBSTITUTED PYRAZOLE COMPOUNDS CONTAINING PYRIMIDINE, THE PREPARATION AND APPLICATION THEREOF Shenyang Sinochem Agrochemicals R&D Co., Ltd. (CN) 2020-09-02 EP disclosed
EP-3299366-A1 SUBSTITUTED PYRAZOLE COMPOUNDS CONTAINING PYRIMIDINE AND PREPARATION METHOD AND USE THEREOF Shenyang Sinochem Agrochemicals R & D Co., Ltd. (CN) 2018-03-28 EP disclosed
WO-2015068773-A1 NITROGEN-CONTAINING SATURATED HETEROCYCLIC COMPOUND 石原産業株式会社 2015-05-14 WO disclosed
EP-0880505-A1 ACYLATED 4-AMINO- AND 4-HYDRAZINOPYRIMIDINES AND THEIR USE AS PESTICIDES BAYER AG (DE) 1998-12-02 EP disclosed
WO-1997028133-A1 ACYLATED 4-AMINO- AND 4-HYDRAZINOPYRIMIDINES AND THEIR USE AS PESTICIDES BAYER AKTIENGESELLSCHAFT (DE) 1997-08-07 WO disclosed
EP-0370391-B1 Process for the preparation of 4,5-dichloro-6-ethyl pyrimidine LONZA AG (CH) 1994-11-02 EP disclosed
US-4977264-A Condensing 2-chloro-3-oxo-pentanoic acid ester with formamidinium salt, reacting with phosphoryl chloride LONZA LTD. (CH) 1990-12-11 US disclosed
EP-0370391-A2 Process for the preparation of 4,5-dichloro-6-ethyl pyrimidine LONZA AG (CH) 1990-05-30 EP disclosed