SCHEMBL8672153

SCHEMBL8672153

CCCCN(C(=O)CCl)c1nc[nH]c(=O)c1Cc1ccc(-c2ccccc2C(=O)OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 2/20 0.47
ACHE P22303 1/20 0.41
AGTR1 P30556 4/20 0.41
AGTR2 P50052 2/20 0.41
BDKRB1 P46663 3/20 0.40
SLC6A3 Q01959 2/20 0.39
SLC6A4 P31645 1/20 0.39
BRS3 P32247 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8979783 0.80 AGTR1 (0.48) LTB4R2ACHEAGTR1AGTR2BDKRB1
SCHEMBL8979910 0.78 BRS3 (0.46) LTB4R2ACHEAGTR1AGTR2BDKRB1
SCHEMBL8801579 0.75 AGTR1 (0.44) LTB4R2ACHEAGTR1AGTR2BDKRB1
SCHEMBL8979781 0.75 AGTR1 (0.48) LTB4R2ACHEAGTR1AGTR2BDKRB1
SCHEMBL8979903 0.73 BRS3 (0.47) LTB4R2ACHEAGTR1AGTR2BDKRB1
SCHEMBL8672154 0.71 ACHE (0.47) ACHEAGTR1AGTR2BDKRB1BRS3
SCHEMBL8979760 0.70 AGTR1 (0.49) LTB4R2ACHEAGTR1AGTR2BRS3
SCHEMBL8979880 0.70 AGTR1 (0.49) LTB4R2ACHEAGTR1AGTR2BRS3
SCHEMBL8672211 0.70 AGTR1 (0.49) LTB4R2ACHEAGTR1AGTR2BRS3
SCHEMBL8979750 0.69 AGTR2 (0.55) AGTR1AGTR2BRS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5804583-A Pyrimidinone derivatives fused to nitrogen heterocycles having a II antagonistic activity ISTITUTO LUSO FARMACO D'ITALIA (IT) 1998-09-08 US disclosed