SCHEMBL8555638

SCHEMBL8555638

CC(=O)c1cccc(-c2ccc(OC(CC(C)O)c3cccnc3)cc2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SUCNR1 Q9BXA5 2/20 0.43
VCP P55072 1/20 0.42
KMO O15229 1/20 0.40
FYN P06241 1/20 0.39
ADRB3 P13945 5/20 0.39
ADRB1 P08588 4/20 0.39
ADRB2 P07550 1/20 0.39
KCNA5 P22460 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HTT P42858 1/20 0.39
KCNH2 Q12809 1/20 0.39
FFAR1 O14842 1/20 0.39
KMT2A Q03164 1/20 0.39
PARP10 Q53GL7 1/20 0.38
PARP11 Q9NR21 1/20 0.38
LMNA P02545 1/20 0.38
GAA P10253 1/20 0.38
PTAFR P25105 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551743 0.92 KMO (0.51) SUCNR1KMOADRB3ADRB1ADRB2
SCHEMBL8552914 0.87 CYP17A1 (0.48) FYNKMT2ALMNA
SCHEMBL8554677 0.87 EPHX1 (0.42) ADRB3ADRB1KCNA5FFAR1LMNA
SCHEMBL8552459 0.85 CYP17A1 (0.44) ADRB3ADRB1FFAR1PTAFR
SCHEMBL8552624 0.85 CYP19A1 (0.47) ADRB3ADRB1KCNA5ALDH1A1
SCHEMBL8109544 0.85 SMN1; SMN2 (0.44) ADRB3ADRB1KCNA5HTTKCNH2
SCHEMBL8118264 0.84 DGAT2 (0.39) ADRB3ADRB1ADRB2KCNA5KCNH2
SCHEMBL8118468 0.84 KCNA5 (0.45) SUCNR1ADRB3ADRB1ADRB2KCNA5
SCHEMBL8118689 0.84 KCNA5 (0.48) KCNA5PTAFR
SCHEMBL8123208 0.84 MKNK1 (0.46) ADRB3ADRB1FFAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865431-A2 COMPOUNDS Astra Pharmaceuticals Limited (GB) 1998-09-23 EP disclosed
WO-1997020815-A1 COMPOUNDS ASTRA PHARMACEUTICALS LTD. (GB) 1997-06-12 WO disclosed