SCHEMBL8677255

SCHEMBL8677255

Brc1cccc2c1CN(c1ccccc1)C2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.47
NPC1 O15118 4/20 0.47
RAB9A P51151 4/20 0.47
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
GAA P10253 1/20 0.44
ALDH1A1 P00352 5/20 0.41
KDM4E B2RXH2 3/20 0.41
TRAP1 Q12931 1/20 0.39
ABHD6 Q9BV23 1/20 0.38
TRPA1 O75762 1/20 0.38
LMNA P02545 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TP53 P04637 1/20 0.38
BACE1 P56817 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
EED O75530 1/20 0.35
POLB P06746 1/20 0.35
PKM P14618 1/20 0.35
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28457709 0.84 EED (0.46) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL30466979 0.77 MEN1 (0.67) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL2185054 0.77 MEN1 (0.67) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL8676808 0.74 NPC1 (0.49) MAPTNPC1RAB9AMEN1KMT2A
SCHEMBL21496659 0.73 HDAC11 (0.62) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL2647074 0.71 CARM1 (0.42) TRAP1ABHD6
SCHEMBL9966898 0.71 ABHD6 (0.41) TRAP1ABHD6TRPA1
SCHEMBL23505868 0.70 TRAP1 (0.42) TRAP1ABHD6TRPA1
SCHEMBL629986 0.70 SIGMAR1 (0.46) LMNA
Hydrochloric Acid SCHEMBL2490663 0.69 SIGMAR1 (0.44) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721248-A CALCIUM AGONISTS; TREATING CARDIOVASCULAR DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1998-02-24 US disclosed
US-5545646-A CARDIOVASCULAR DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1996-08-13 US disclosed
EP-0630895-A1 4-Bicyclic substituted dihydropyridines, process for their preparation and their use in medicaments BAYER AG (DE) 1994-12-28 EP disclosed