SCHEMBL8678271

SCHEMBL8678271

COc1ccc(-c2ccc(C)nc2-c2ccc(O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.56
NOX1 Q9Y5S8 1/20 0.52
KMT2A Q03164 5/20 0.49
SYK P43405 3/20 0.48
AURKB Q96GD4 2/20 0.48
INCENP Q9NQS7 2/20 0.48
MAPT P10636 5/20 0.48
TP53 P04637 3/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
HTT P42858 1/20 0.48
MAPK10 P53779 1/20 0.48
PTK2B Q14289 1/20 0.48
NCOA1 Q15788 1/20 0.48
NCOA3 Q9Y6Q9 1/20 0.48
MEN1 O00255 3/20 0.48
NPC1 O15118 1/20 0.48
APP P05067 1/20 0.47
LTA4H P09960 1/20 0.47
HSP90AA1 P07900 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5904242 0.92 KMT2A (0.53) ESR2KMT2ASYKAURKBINCENP
Dimethylamine SCHEMBL5358041 0.89 KMT2A (0.50) KMT2ASYKAURKBINCENPMAPT
Dimethylamine SCHEMBL9695311 0.87 KMT2A (0.49) KMT2ASYKAURKBINCENPMAPT
SCHEMBL8675465 0.84 MAPT (0.59) ESR2NOX1KMT2AMAPTTP53
SCHEMBL4037256 0.83 ALDH1A1 (0.57) ESR2NOX1SYKAURKBINCENP
SCHEMBL8678444 0.81 NPSR1 (0.55) KMT2ASYKAURKBINCENPMAPT
SCHEMBL8811479 0.80 ESR2 (0.51) ESR2NOX1KMT2AMAPTTP53
SCHEMBL8680387 0.79 MAPT (0.56) ESR2NOX1KMT2AMAPTTP53
SCHEMBL8677193 0.78 MAPT (0.52) ESR2NOX1KMT2AMAPTTP53
SCHEMBL8809606 0.78 ESR1 (0.48) ESR2KMT2AMAPTTP53MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750708-A Pyridine compounds intermediates processes compositions and methods ELI LILLY AND COMPANY (US) 1998-05-12 US disclosed
US-5672609-A POSTMENOPAUSAL SYNDROME; ANTILIPEMIC AND -CARCINOGENIC AGENTS; OSTEOPOROSIS; CARDIOTONIC AGENTS; RESTENOSIS; SIDE EFFECT REDUCTION COMPARED TO ESTROGEN ELI LILLY AND COMPANY (US) 1997-09-30 US disclosed
WO-1997004778-A1 PYRIDINE COMPOUNDS, INTERMEDIATES, PROCESSES, COMPOSITIONS, AND METHODS ELI LILLY AND COMPANY (US) 1997-02-13 WO disclosed