SCHEMBL8678977

SCHEMBL8678977

CC(C)(N=C=O)c1cccc(C(C)(C)N=C=O)c1.CCCCCCCN=C=O.CCCCCN=C=O

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NAAA Q02083 1/20 0.34
SCN5A Q14524 3/20 0.33
SCN9A Q15858 3/20 0.33
HDAC3 O15379 2/20 0.30
HDAC1 Q13547 2/20 0.30
HDAC2 Q92769 2/20 0.30
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7732599 0.90 NAAA (0.35) NAAA
SCHEMBL34924 0.80 ESR1 (0.36) HDAC2
SCHEMBL11305988 0.77 KIF11 (0.37) NAAACNR1CNR2
SCHEMBL11646108 0.77 NAAA (0.47) NAAA
SCHEMBL14094919 0.76 NPC1 (0.41)
Carbimide SCHEMBL4253887 0.75 ESR1 (0.33) HDAC2
SCHEMBL12050426 0.75 ESR1 (0.33) HDAC2
SCHEMBL2494913 0.75 ESR1 (0.33) HDAC2
SCHEMBL39076 0.75 HDAC8 (0.43) HDAC3HDAC2
SCHEMBL24833769 0.74 PGK1 (0.32) HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880558-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED INDANE LIBRARIES ELI LILLY AND COMPANY (US) 1998-12-02 EP disclosed
WO-1997026300-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED INDANE LIBRARIES ELI LILLY AND COMPANY (US) 1997-07-24 WO disclosed