SCHEMBL8683080

SCHEMBL8683080

CC(=O)Nc1c(C)ccnc1C=NNC(N)=S

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RRM2 P31350 7/20 0.50
NCOA3 Q9Y6Q9 3/20 0.50
NCOA1 Q15788 2/20 0.50
RRM1 P23921 1/20 0.50
RRM2B Q7LG56 1/20 0.50
CISD1 Q9NZ45 1/20 0.50
G6PD P11413 1/20 0.45
CTH P32929 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1882894 0.79 RRM2 (0.61) RRM2NCOA3NCOA1RRM1RRM2B
SCHEMBL8684404 0.79 RRM2 (0.57) RRM2NCOA3NCOA1RRM1RRM2B
SCHEMBL29569419 0.79 RRM2 (0.61) RRM2NCOA3NCOA1RRM1RRM2B
SCHEMBL1882892 0.79 RRM2 (0.61) RRM2NCOA3NCOA1RRM1RRM2B
SCHEMBL8682963 0.74 NCOA3 (0.46) RRM2NCOA3NCOA1RRM1RRM2B
SCHEMBL1904117 0.72 RRM2 (0.70) RRM2NCOA3NCOA1RRM1RRM2B
SCHEMBL8683501 0.70 RRM2 (0.48) RRM2NCOA3NCOA1G6PDKDM4E
SCHEMBL16919139 0.70 ALDH1A1 (0.49) KDM4EALDH1A1CYP1A2
SCHEMBL6261110 0.69 RRM2 (0.71) RRM2NCOA3NCOA1CTHKDM4E
SCHEMBL6261112 0.69 RRM2 (0.71) RRM2NCOA3NCOA1CTHKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721259-A Method of using 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1998-02-24 US disclosed
EP-0570294-B1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents UNIV YALE (US) 1997-07-30 EP disclosed
US-5281715-A 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1994-01-25 US disclosed
EP-0570294-A1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents YALE UNIVERSITY (US) 1993-11-18 EP disclosed