SCHEMBL8683408

SCHEMBL8683408

Oc1ccc(N2CCN(c3ccncc3)CC2)c(-c2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHKA P35790 1/20 0.45
METAP1 P53582 1/20 0.42
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
ALOX5 P09917 1/20 0.40
CSNK1D P48730 2/20 0.40
MAPK14 Q16539 2/20 0.40
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
KHK P50053 1/20 0.39
USP2 O75604 1/20 0.39
CYP3A4 P08684 1/20 0.39
PIK3CA P42336 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8681378 0.77 CHKA (0.46) CHKAMAPTKDM4EGAASMN1; SMN2
SCHEMBL7401781 0.75 HRH3 (0.51) MAPTSMN1; SMN2
SCHEMBL7401777 0.74 PPARG (0.45) SMN1; SMN2MEN1ALDH1A1KMT2A
SCHEMBL7334978 0.73 CHKA (0.61) CHKAMAPTKDM4EGAASMN1; SMN2
SCHEMBL18590696 0.73 CHKA (0.67) CHKAMAPTKDM4EGAACA12
SCHEMBL8636540 0.72 GAA (0.62) CHKAMAPTKDM4EGAACA12
SCHEMBL7398706 0.72 DRD2 (0.55) CHKAMAPTKDM4EGAAKHK
SCHEMBL7330427 0.72 PPARG (0.45)
SCHEMBL28302485 0.72 HSD17B10 (0.43) ALOX5USP2MEN1ALDH1A1KMT2A
SCHEMBL1424248 0.72 ALOX5 (0.59) MAPTALOX5MAPK14SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed