SCHEMBL8685294

SCHEMBL8685294

CC(=O)Oc1c(C)ccnc1C(OC(C)=O)OC(C)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.41
HSD17B10 Q99714 2/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
PTPN1 P18031 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTT P42858 2/20 0.36
TP53 P04637 1/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
ELANE P08246 1/20 0.34
LMNA P02545 2/20 0.33
TSHR P16473 2/20 0.33
PDE4A P27815 2/20 0.33
ABCB11 O95342 1/20 0.33
ESR1 P03372 1/20 0.33
CYP3A4 P08684 1/20 0.33
ADRA2A P08913 1/20 0.33
CYP2C9 P11712 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17706563 0.73 KDM4E (0.45) KDM4EHSD17B10ALDH1A1HPGDPTPN1
SCHEMBL27693258 0.70 HSD17B10 (0.41) KDM4EHSD17B10ALDH1A1HPGDPTPN1
SCHEMBL16265058 0.69 KDM4E (0.59) KDM4EHSD17B10ALDH1A1HPGDPTPN1
SCHEMBL8685106 0.69 ALDH1A1 (0.41) KDM4EHSD17B10ALDH1A1HPGDPTPN1
SCHEMBL9693906 0.68 TDP1 (0.48) KDM4EHSD17B10ALDH1A1HPGDHTT
SCHEMBL27465233 0.66 NOS3 (0.41) KDM4EHSD17B10ALDH1A1HPGDPTPN1
SCHEMBL2059537 0.66 KDM4E (0.71) KDM4EHSD17B10ALDH1A1HPGDPTPN1
SCHEMBL5865887 0.65 KDM4E (0.41) KDM4EHSD17B10ALDH1A1HPGDHTT
SCHEMBL16450253 0.64 KDM4E (0.53) KDM4EHSD17B10ALDH1A1HPGDPTPN1
SCHEMBL15174454 0.64 NOS3 (0.39) KDM4EALDH1A1SMN1; SMN2HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721259-A Method of using 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1998-02-24 US disclosed
EP-0570294-B1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents UNIV YALE (US) 1997-07-30 EP disclosed
US-5281715-A 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1994-01-25 US disclosed
EP-0570294-A1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents YALE UNIVERSITY (US) 1993-11-18 EP disclosed