SCHEMBL8686276

SCHEMBL8686276

FC(F)(F)c1ccc(OCCc2ncc[nH]2)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 4/20 0.46
TAAR1 Q96RJ0 1/20 0.43
LTA4H P09960 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP19A1 P11511 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
MAOB P27338 4/20 0.39
DRD2 P14416 1/20 0.39
DRD1 P21728 1/20 0.39
DRD3 P35462 1/20 0.39
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
HMOX1 P09601 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8685451 0.93 NOS1 (0.47) NOS1TAAR1LTA4HCYP1A2CYP3A4
SCHEMBL11760748 0.84 MAOB (0.47) NOS1TAAR1MAOBHMOX1
SCHEMBL8635977 0.80 LTA4H (0.44) LTA4HCYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL28261194 0.80 TAAR1 (0.46) TAAR1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL6181232 0.80 NPC1 (0.49) TAAR1CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL8684972 0.80 FPR2 (0.43) NOS1TAAR1CYP1A2CYP3A4CYP2D6
SCHEMBL8690250 0.80 HRH3 (0.48) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL11581355 0.79 TAAR1 (0.53) TAAR1LTA4HCYP1A2CYP3A4CYP2D6
SCHEMBL8684911 0.78 CYP1A2 (0.45) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL8685448 0.77 CYP1A2 (0.48) TAAR1LTA4HCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5708171-A HISTAMINE H3-RECEPTOR ANTAGONIST INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 1998-01-13 US claimed
US-5708171-A HISTAMINE H3-RECEPTOR ANTAGONIST INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 1998-01-13 US disclosed