SCHEMBL8689010

SCHEMBL8689010

NS(=O)(=O)c1ccccc1-n1nc(C(F)(F)F)cc1-c1ccco1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 9/20 0.47
PTGS1 P23219 5/20 0.46
PDPK1 O15530 4/20 0.45
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8637761 0.82 PTGS2 (0.48) PTGS2PTGS1PDPK1
SCHEMBL8637022 0.82 PTGS2 (0.47) PTGS2PTGS1PDPK1
SCHEMBL8635874 0.82 PTGS2 (0.48) PTGS2PTGS1PDPK1
SCHEMBL8640768 0.82 PTGS2 (0.67) PTGS2PTGS1PDPK1TSHR
SCHEMBL6343163 0.81 PTGS2 (0.67) PTGS2PTGS1PDPK1TSHR
SCHEMBL8637585 0.80 PDPK1 (0.69) PTGS2PTGS1PDPK1TSHR
SCHEMBL8639323 0.80 PTGS2 (0.51) PTGS2PTGS1PDPK1
SCHEMBL8637765 0.80 PDPK1 (0.50) PTGS2PTGS1PDPK1
SCHEMBL950629 0.80 RXRA (0.52) PTGS2PTGS1KDM4EALDH1A1HPGD
SCHEMBL7237134 0.80 KDM4E (0.42) PTGS2PTGS1PDPK1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed
US-5510496-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1996-04-23 US disclosed
US-5504215-A Substituted pyrazolyl benzenesulfonamide compounds for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-04-02 US disclosed