SCHEMBL8690929

SCHEMBL8690929

N#Cc1nn(-c2ccccc2S(N)(=O)=O)c(-c2ccc(F)cc2)c1Cl

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.54
PTGS1 P23219 7/20 0.54
CA2 P00918 3/20 0.39
CA7 P43166 2/20 0.39
CNR1 P21554 6/20 0.37
F10 P00742 2/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA9 Q16790 1/20 0.35
LMNA P02545 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CA4 P22748 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689215 0.91 PTGS2 (0.65) PTGS2PTGS1CA2CA7CNR1
SCHEMBL8689138 0.91 PTGS2 (0.55) PTGS2PTGS1CA2CA7F10
SCHEMBL8689036 0.87 PTGS2 (0.40) PTGS2PTGS1CA2CA7CNR1
SCHEMBL6345546 0.80 PTGS2 (0.83) PTGS2PTGS1CA2CA1CA9
SCHEMBL8691576 0.77 CA2 (0.41) PTGS2PTGS1CA2CA7CNR1
SCHEMBL8693265 0.75 PTGS2 (0.52) PTGS2PTGS1CA2CA7F10
SCHEMBL8693252 0.75 PTGS2 (0.65) PTGS2PTGS1CA2CA12CA1
SCHEMBL8422281 0.74 PTGS1 (0.44) PTGS2PTGS1CA2CA7CNR1
SCHEMBL8421921 0.74 CA2 (0.44) PTGS2PTGS1CA2CA7CNR1
SCHEMBL7059987 0.73 PTGS2 (0.47) PTGS2PTGS1CA2CA7F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed