SCHEMBL8694236

SCHEMBL8694236

CCCCNC(=S)Nc1nn(Cc2ccccc2)cc1C(=O)OCC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
KMT2A Q03164 3/20 0.46
MEN1 O00255 2/20 0.46
GAA P10253 2/20 0.46
MAPT P10636 2/20 0.46
ALOX12 P18054 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
RXFP1 Q9HBX9 1/20 0.45
LMNA P02545 2/20 0.45
SIRT5 Q9NXA8 5/20 0.45
HTT P42858 2/20 0.43
AGTR1 P30556 1/20 0.41
KDM4E B2RXH2 1/20 0.41
CREBBP Q92793 1/20 0.41
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
DGAT1 O75907 1/20 0.41
P2RX7 Q99572 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8693140 0.96 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1GAAMAPT
SCHEMBL8695938 0.94 ALDH1A1 (0.47) ALDH1A1KMT2AMEN1GAAMAPT
SCHEMBL8696343 0.90 ALDH1A1 (0.47) ALDH1A1GAAMAPTRAB9ASMN1; SMN2
SCHEMBL8692678 0.89 HTT (0.46) ALDH1A1KMT2AGAAMAPTALOX12
SCHEMBL8698640 0.87 ALDH1A1 (0.41) ALDH1A1KMT2AMEN1GAAMAPT
SCHEMBL8696191 0.86 EPHX1 (0.47) ALDH1A1KMT2AGAARAB9ALMNA
SCHEMBL8699774 0.86 ALDH1A1 (0.43) ALDH1A1KMT2AMEN1GAAMAPT
SCHEMBL8693986 0.86 ALDH1A1 (0.43) ALDH1A1KMT2AMEN1GAAMAPT
SCHEMBL8696777 0.85 POLB (0.44) ALDH1A1KMT2AMEN1MAPTLMNA
SCHEMBL8698769 0.84 ALDH1A1 (0.45) ALDH1A1NPC1RAB9ASMN1; SMN2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849779-A Pyrazole derivatives and their pharmaceutical use JAPAN ENERGY CORPORATION (JP) 1998-12-15 US disclosed
EP-0810217-A1 Pyrazole derivatives and their pharmaceutical use as smooth muscle cell growth inhibitors JAPAN ENERGY CORPORATION (JP) 1997-12-03 EP disclosed