SCHEMBL8696191

SCHEMBL8696191

CCCCCCNC(=O)Nc1nn(Cc2ccccc2)cc1C(=O)OCC

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 7/20 0.47
ALDH1A1 P00352 4/20 0.47
HTT P42858 2/20 0.47
LMNA P02545 1/20 0.45
CREBBP Q92793 1/20 0.43
POLB P06746 1/20 0.42
KDM4E B2RXH2 2/20 0.42
TSHR P16473 2/20 0.42
GAA P10253 1/20 0.42
RAB9A P51151 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
AGTR1 P30556 1/20 0.41
KLKB1 P03952 1/20 0.41
KMT2A Q03164 1/20 0.41
DGAT1 O75907 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696343 0.96 ALDH1A1 (0.47) EPHX1ALDH1A1HTTLMNACREBBP
SCHEMBL8593357 0.92 ALDH1A1 (0.48) ALDH1A1HTTLMNACREBBPPOLB
SCHEMBL8693140 0.90 ALDH1A1 (0.45) ALDH1A1LMNACREBBPPOLBKDM4E
SCHEMBL8696100 0.89 EPHX1 (0.52) EPHX1ALDH1A1HTTCREBBPPOLB
SCHEMBL8693552 0.87 MAPT (0.54) ALDH1A1LMNAPOLBKDM4ETSHR
SCHEMBL8695984 0.87 EPHX1 (0.42) EPHX1ALDH1A1HTTKDM4ETSHR
SCHEMBL8694236 0.86 ALDH1A1 (0.46) ALDH1A1HTTLMNACREBBPKDM4E
SCHEMBL8698725 0.86 EPHX1 (0.41) EPHX1ALDH1A1HTTKDM4ETSHR
SCHEMBL8693110 0.86 EPHX1 (0.41) EPHX1ALDH1A1HTTKDM4ETSHR
SCHEMBL8696177 0.84 ALDH1A1 (0.46) EPHX1ALDH1A1HTTCREBBPPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849779-A Pyrazole derivatives and their pharmaceutical use JAPAN ENERGY CORPORATION (JP) 1998-12-15 US disclosed
EP-0810217-A1 Pyrazole derivatives and their pharmaceutical use as smooth muscle cell growth inhibitors JAPAN ENERGY CORPORATION (JP) 1997-12-03 EP disclosed