SCHEMBL8695151

SCHEMBL8695151

OCc1ccc(OCc2ccccc2)c(Br)n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP28 Q96RU2 1/20 0.43
USP25 Q9UHP3 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
RAB9A P51151 1/20 0.43
HTT P42858 2/20 0.42
ATP4A P20648 1/20 0.42
ATP4B P51164 1/20 0.42
LIPE Q05469 1/20 0.41
FOLH1 Q04609 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MAPT P10636 1/20 0.41
MAPK1 P28482 1/20 0.41
LTA4H P09960 1/20 0.41
MAPK14 Q16539 1/20 0.41
CCR5 P51681 2/20 0.40
PTGER1 P34995 1/20 0.40
BRD4 O60885 1/20 0.40
STAT3 P40763 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8694874 0.85 CNR1 (0.41) RHEB
SCHEMBL17536018 0.83 S1PR4 (0.52) SMN1; SMN2RAB9AATP4AATP4BLIPE
SCHEMBL2904391 0.83 ATP4A (0.43) SMN1; SMN2RAB9AHTTATP4AATP4B
SCHEMBL2026551 0.81 SMN1; SMN2 (0.54) SMN1; SMN2HTTATP4AATP4BLIPE
SCHEMBL8694664 0.81 S1PR4 (0.51) SMN1; SMN2RAB9AHTTATP4AATP4B
Hydrochloric Acid SCHEMBL11833848 0.80 SMN1; SMN2 (0.52) SMN1; SMN2HTTATP4AATP4BLIPE
SCHEMBL2435879 0.79 L3MBTL1 (0.44) SMN1; SMN2RAB9AHTTLIPEFOLH1
SCHEMBL24930498 0.78 MPO (0.50) SMN1; SMN2RAB9AHTTATP4AATP4B
SCHEMBL22850860 0.78 MAPT (0.43) SMN1; SMN2RAB9AHTTFOLH1TDP1
SCHEMBL31394965 0.76 SMN1; SMN2 (0.50) SMN1; SMN2RAB9AHTTLIPEFOLH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726315-A Certain 3-hydroxy-6-hydroxymethyl-pyridine intermediates SMITHKLINE BEECHAM PLC (GB) 1998-03-10 US disclosed
US-5646286-A Palladium catalyzed vinylic substitution reactions with 2-substituted-pyridines SMITHKLINE BEECHAM PLC (GB) 1997-07-08 US disclosed
EP-0705249-B1 PALLADIUM CATALYZED VINYLIC SUBSTITUTION REACTIONS WITH 2-SUBSTITUTED-PYRIDINES SMITHKLINE BEECHAM PLC (GB) 1997-05-14 EP disclosed
EP-0705249-A1 PALLADIUM CATALYZED VINYLIC SUBSTITUTION REACTIONS WITH 2-SUBSTITUTED-PYRIDINES SMITHKLINE BEECHAM PLC (GB) 1996-04-10 EP disclosed
WO-1995000487-A1 PALLADIUM CATALYZED VINYLIC SUBSTITUTION REACTIONS WITH 2-SUBSTITUTED-PYRIDINES SMITHKLINE BEECHAM PLC (GB) 1995-01-05 WO disclosed