SCHEMBL8696358

SCHEMBL8696358

CCOC(=O)Oc1[nH]c2c3ccccc3n(C)c2c1-c1ccc2c(c1)CCO2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK1 P49759 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
FABP4 P15090 7/20 0.37
KDM4E B2RXH2 3/20 0.36
KMT2A Q03164 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
ALDH1A1 P00352 3/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
FABP3 P05413 3/20 0.35
FABP5 Q01469 2/20 0.35
PKM P14618 1/20 0.35
CHRM5 P08912 4/20 0.34
CHRM1 P11229 4/20 0.34
CHRM4 P08173 2/20 0.34
CHRM3 P20309 2/20 0.34
CHRM2 P08172 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8696580 0.79 ALDH1A1 (0.46) KDM4EKMT2AALDH1A1SMN1; SMN2POLB
SCHEMBL8697497 0.78 L3MBTL1 (0.48) NPC1RAB9AL3MBTL1KMT2ASMN1; SMN2
SCHEMBL8551756 0.76 CLK1 (0.45) CLK1NPC1RAB9AFABP4KDM4E
SCHEMBL8552505 0.74 CLK1 (0.44) CLK1NPC1RAB9AFABP4KDM4E
SCHEMBL8702719 0.73 ALDH1A1 (0.41) L3MBTL1KDM4EKMT2ARXFP1ALDH1A1
SCHEMBL8547598 0.73 NPC1 (0.40) CLK1NPC1RAB9AFABP4KDM4E
SCHEMBL8546890 0.73 EDNRB (0.44) CLK1NPC1RAB9AFABP4KDM4E
SCHEMBL8697402 0.73 NTRK1 (0.39) L3MBTL1KDM4EKMT2AALDH1A1HPGD
SCHEMBL8552118 0.72 NPC1 (0.42) CLK1NPC1RAB9AFABP4KDM4E
SCHEMBL8552363 0.72 NPC1 (0.41) CLK1NPC1RAB9AFABP4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998042709-A1 ENDOTHELIN-RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 1998-10-01 WO disclosed