SCHEMBL8698699

SCHEMBL8698699

O=C(Nc1ccccc1)Nc1nn(Cc2ccccc2)cc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 7/20 0.58
ADORA2B P29275 3/20 0.58
ADORA1 P30542 3/20 0.58
ALDH1A1 P00352 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
ADORA2A P29274 2/20 0.46
TP53 P04637 2/20 0.45
EPHX1 P07099 1/20 0.45
TSHR P16473 1/20 0.45
EPHX2 P34913 1/20 0.45
CDK9 P50750 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
KMT2A Q03164 2/20 0.45
PPIA P62937 1/20 0.44
NPC1 O15118 1/20 0.43
POLB P06746 1/20 0.43
RAB9A P51151 1/20 0.43
GRIK1 P39086 1/20 0.43
MAOA P21397 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8693785 0.86 ADORA3 (0.53) ADORA3ADORA2BADORA1ALDH1A1ADORA2A
SCHEMBL8698039 0.85 ADORA3 (0.52) ADORA3ADORA2BADORA1ALDH1A1L3MBTL1
SCHEMBL6312199 0.84 ALDH1A1 (0.50) ADORA3ADORA2BADORA1ALDH1A1L3MBTL1
SCHEMBL8695495 0.83 L3MBTL1 (0.45) ADORA3ADORA2BADORA1ALDH1A1L3MBTL1
SCHEMBL8696177 0.81 ALDH1A1 (0.46) ADORA3ADORA2BADORA1ALDH1A1L3MBTL1
SCHEMBL8693738 0.80 HPGD (0.52) ALDH1A1TP53EPHX1TSHREPHX2
SCHEMBL8696100 0.79 EPHX1 (0.52) ALDH1A1L3MBTL1EPHX1EPHX2SMN1; SMN2
SCHEMBL28764370 0.77 ALDH1A1 (0.49) ADORA3ADORA2BADORA1ALDH1A1L3MBTL1
SCHEMBL8696733 0.76 KMT2A (0.46) ADORA3ALDH1A1L3MBTL1SMN1; SMN2KMT2A
SCHEMBL8692678 0.74 HTT (0.46) ALDH1A1L3MBTL1TSHRSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5849779-A Pyrazole derivatives and their pharmaceutical use JAPAN ENERGY CORPORATION (JP) 1998-12-15 US disclosed
EP-0810217-A1 Pyrazole derivatives and their pharmaceutical use as smooth muscle cell growth inhibitors JAPAN ENERGY CORPORATION (JP) 1997-12-03 EP disclosed