SCHEMBL8699190

SCHEMBL8699190

CN(C)c1ccc(C=O)c2ccccc12.O=Cc1cccc(F)c1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RET P07949 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
FLT3 P36888 1/20 0.40
ERN1 O75460 1/20 0.39
CHEK1 O14757 1/20 0.39
NEK2 P51955 1/20 0.39
LIMK1 P53667 1/20 0.39
DYRK1A Q13627 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
EP300 Q09472 1/20 0.38
KAT2B Q92831 1/20 0.38
KAT8 Q9H7Z6 1/20 0.38
KDM4E B2RXH2 2/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35
CA2 P00918 1/20 0.35
LMNA P02545 3/20 0.34
MAPT P10636 2/20 0.34
POLB P06746 1/20 0.34
NFKB1 P19838 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29708057 0.84 CHEK1 (0.52) RETTDP1FLT3CHEK1NEK2
SCHEMBL346454 0.84 CHEK1 (0.52) RETTDP1FLT3CHEK1NEK2
SCHEMBL13486828 0.81 CA2 (0.49) RETTDP1FLT3CHEK1NEK2
SCHEMBL11895872 0.77 NFE2L2 (0.53) RETTDP1CHEK1NEK2LIMK1
SCHEMBL29403281 0.77 NFE2L2 (0.53) RETTDP1CHEK1NEK2LIMK1
SCHEMBL11895869 0.77 NFE2L2 (0.53) RETTDP1CHEK1NEK2LIMK1
SCHEMBL154794 0.76 ERN1 (0.61) TDP1ERN1LMNAHTTSMN1; SMN2
SCHEMBL12143561 0.72 ERN1 (0.57) TDP1ERN1KDM4ELMNAHTT
Hydrazine SCHEMBL27868863 0.72 ERN1 (0.57) TDP1ERN1LMNAALDH1A1MEN1
SCHEMBL9671258 0.72 ERN1 (0.57) TDP1ERN1KDM4ELMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998008813-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED PYRROLIDINE LIBRARIES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed