SCHEMBL8699298

SCHEMBL8699298

CC(=O)NCc1ccc(C(=O)NC(=N)N)cc1-n1cccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.46
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2C9 P11712 1/20 0.43
SETDB1 Q15047 3/20 0.38
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AOC2 O75106 2/20 0.36
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
MAPT P10636 2/20 0.34
POLB P06746 1/20 0.34
RECQL P46063 1/20 0.34
BLM P54132 1/20 0.34
MCL1 Q07820 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8705215 0.96 NQO2 (0.45) NQO2CYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL8699878 0.84 AOC2 (0.40) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1
SCHEMBL8707021 0.81 AOC2 (0.36) CYP1A2CYP3A4CYP2C19ALDH1A1SMN1; SMN2
SCHEMBL8700249 0.81 PLK1 (0.37) CYP1A2CYP3A4CYP2C19ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL8703965 0.81 SPHK1 (0.38) CYP1A2CYP3A4CYP2C19ALDH1A1SMN1; SMN2
Guanidine SCHEMBL8705211 0.80 CYP1A2 (0.40) NQO2CYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL7816932 0.80 CYP1A2 (0.43) CYP1A2CYP3A4CYP2C19CYP2C9SETDB1
SCHEMBL7825259 0.79 CYP1A2 (0.47) NQO2CYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL8705218 0.79 CYP1A2 (0.37) NQO2CYP1A2CYP3A4CYP2C19CYP2C9
SCHEMBL8703469 0.79 LMNA (0.40) CYP1A2CYP3A4CYP2C19CYP2C9ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5824691-A CARDIOVASCULAR, CEREBROVASCULAR, RENAL DISEASES; SHOCK, ARTERIOSCLEROSIS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-10-20 US disclosed