SCHEMBL8700537

SCHEMBL8700537

N#Cc1ccc(C(c2cncnc2)c2cc3ccccc3o2)c(F)c1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 12/20 0.47
CYP2A6 P11509 1/20 0.36
CYP26A1 O43174 2/20 0.33
MAPT P10636 1/20 0.32
KCNH2 Q12809 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP3A5 P20815 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
S1PR1 P21453 1/20 0.31
S1PR3 Q99500 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8702186 0.88 CYP19A1 (0.47) CYP19A1CYP2A6CYP26A1MAPT
SCHEMBL8697486 0.85 CYP19A1 (0.46) CYP19A1CYP26A1CYP3A4
SCHEMBL8697788 0.83 CYP19A1 (0.60) CYP19A1CYP2A6CYP26A1MAPT
SCHEMBL8700262 0.79 CYP19A1 (0.42) CYP19A1KCNH2CYP3A4
SCHEMBL8702245 0.75 CYP19A1 (0.72) CYP19A1CYP26A1CYP3A4
SCHEMBL8697118 0.74 CYP19A1 (0.55) CYP19A1CYP26A1MAOAMAOB
SCHEMBL8697624 0.74 CYP19A1 (0.50) CYP19A1CYP2A6CYP26A1MAPT
SCHEMBL8699998 0.74 CYP26A1 (0.44) CYP19A1CYP26A1
SCHEMBL8696314 0.72 CYP19A1 (0.41) CYP19A1CYP2A6MAPTKCNH2CYP3A4
SCHEMBL8700871 0.72 CYP3A4 (0.43) CYP19A1CYP2A6MAPTKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018791-A1 HETEROCYCLIC FURAN COMPOUNDS, THEIR PREPARATION AND USE AS AROMATASE INHIBITORS A. MENARINI INDUSTRIE FARMACEUTICHE RIUNITE S.R.L. (IT) 1998-05-07 WO claimed