SCHEMBL8700703

SCHEMBL8700703

O=C(O)c1ccc(-c2cc[nH]n2)c([N+](=O)[O-])c1

nearest known ligand 0.54

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.54
LMNA P02545 1/20 0.54
TSHR P16473 2/20 0.50
HCAR3 P49019 13/20 0.47
APEX1 P27695 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11195885 0.80 CASP6 (0.75) CASP6LMNATSHRHCAR3APEX1
SCHEMBL8809569 0.80 MAPT (0.52) TSHR
SCHEMBL30978366 0.77 CASP6 (0.57) CASP6LMNATSHRHCAR3APEX1
SCHEMBL31548567 0.76 CASP6 (0.64) CASP6LMNATSHRHCAR3APEX1
SCHEMBL17197945 0.76 CASP6 (0.68) CASP6LMNATSHRHCAR3APEX1
SCHEMBL30978367 0.75 ALDH1A1 (0.60) CASP6LMNATSHRHCAR3
SCHEMBL11761567 0.75 ALDH1A1 (0.60) CASP6LMNATSHRHCAR3
SCHEMBL31174723 0.74 ALDH1A1 (0.50) LMNA
SCHEMBL2062065 0.74 ALDH1A1 (0.50) LMNA
SCHEMBL9557826 0.74 CASP6 (0.66) CASP6LMNATSHRHCAR3APEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5834471-A Amide derivatives as 5HT1D receptor antagonists SMITHKLINE BEECHAM P.L.C. (GB) 1998-11-10 US disclosed
EP-0712397-A1 AMIDE DERIVATIVES AS 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1996-05-22 EP disclosed
WO-1995004729-A1 AMIDE DERIVATIVES AS 5HT1D RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM PLC (GB) 1995-02-16 WO disclosed