SCHEMBL8705223

SCHEMBL8705223

COC(=O)c1cc(S(C)(=O)=O)c(-n2cc(C)nc2C)cc1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.37
NR3C2 P08235 1/20 0.37
ILK Q13418 1/20 0.36
PKM P14618 1/20 0.36
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
NR1H2 P55055 5/20 0.34
NR1H3 Q13133 4/20 0.34
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
SDHB P21912 1/20 0.32
KDM4E B2RXH2 1/20 0.32
KMT2A Q03164 1/20 0.32
F10 P00742 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8702046 0.86 KDM4E (0.39) ALDH1A1HPGDTSHRHSD17B10MAPT
SCHEMBL8705953 0.86 NR1I2 (0.40) ALDH1A1HPGDTSHRHSD17B10MAPT
SCHEMBL8705762 0.85 SDHB (0.37) PKMALDH1A1MAPTNR1H2NR1H3
SCHEMBL8705360 0.85 MAPT (0.33) NR3C1NR3C2ALDH1A1HSD17B10MAPT
SCHEMBL8703753 0.85 NR3C1 (0.33) NR3C1NR3C2MAPTNPSR1NR1H2
SCHEMBL8706166 0.85 MAPT (0.34) NR3C1NR3C2MAPTNPSR1NR1H2
SCHEMBL8699344 0.84 GAA (0.42) ALDH1A1HPGDMAPTNPSR1PIK3CD
SCHEMBL8704804 0.84 MAPT (0.33) NR3C1NR3C2ALDH1A1HPGDMAPT
SCHEMBL8705210 0.82 VCAM1 (0.45) MAPTKDM4EKMT2A
SCHEMBL8703808 0.81 NR3C2 (0.40) NR3C2PKMALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753680-A Heterocyclyl-benzoylguanidines MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-05-19 US disclosed