SCHEMBL8708554

SCHEMBL8708554

COC(=O)CC[C@H]1CCC[C@H](COS(C)(=O)=O)O1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.33
CA14 Q9ULX7 1/20 0.33
TSHR P16473 2/20 0.32
EPHX2 P34913 2/20 0.32
SIRT2 Q8IXJ6 1/20 0.31
LMNA P02545 2/20 0.31
ALDH1A1 P00352 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
POLB P06746 1/20 0.31
HCRTR2 O43614 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8708555 1.00 CA12 (0.33) CA12CA14TSHREPHX2SIRT2
SCHEMBL8708864 0.79 TSHR (0.39) CA12CA14TSHREPHX2SIRT2
SCHEMBL8708861 0.79 TSHR (0.39) CA12CA14TSHREPHX2SIRT2
SCHEMBL8784357 0.76 FKBP1A (0.35) TSHREPHX2SIRT2ALDH1A1
SCHEMBL8784352 0.76 FKBP1A (0.35) TSHREPHX2SIRT2ALDH1A1
SCHEMBL12869959 0.75 KDM4E (0.37) TSHRLMNAALDH1A1
SCHEMBL8710178 0.74 MIF (0.32)
SCHEMBL8708552 0.73 TRPA1 (0.32) CA14LMNA
SCHEMBL8711480 0.72 ACHE (0.31) TSHRLMNAALDH1A1
SCHEMBL8710648 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5736549-A INHIBITORS OF PURINE NUCLEOSIDE PHOSPHORYLASE, USED FOR TREATING OR PREVENTING TISSUE REJECTION OR SELECTIVE SUPPRESSION OF MAMMALIAN T-CELL FUNCTION CHIROSCIENCE LIMITED (GB) 1998-04-07 US disclosed
EP-0784624-A1 PURINE AND GUANINE COMPOUNDS AS INHIBITORS OF PNP Chiroscience Limited (GB) 1997-07-23 EP disclosed
WO-1996011200-A1 PURINE AND GUANINE COMPOUNDS AS INHIBITORS OF PNP CHIROSCIENCE LIMITED (GB) 1996-04-18 WO disclosed