SCHEMBL8709208

SCHEMBL8709208

CC(C(=O)O)N(C(=O)OC(C)(C)C)c1ccc2ncccc2c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX15 P16050 1/20 0.42
HTT P42858 1/20 0.42
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
ALDH1A1 P00352 5/20 0.40
PABPC1 P11940 1/20 0.40
PLK1 P53350 1/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
LMNA P02545 1/20 0.39
CYP3A4 P08684 1/20 0.39
NPC1 O15118 4/20 0.39
POLB P06746 3/20 0.39
MEN1 O00255 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
DOT1L Q8TEK3 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
RAB9A P51151 3/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709207 1.00 ALOX15 (0.42) ALOX15HTTAKR1C3AKR1C2ALDH1A1
SCHEMBL1325516 0.84 MEN1 (0.43) AKR1C3AKR1C2ALDH1A1SMN1; SMN2MEN1
SCHEMBL995191 0.84 MEN1 (0.43) AKR1C3AKR1C2ALDH1A1SMN1; SMN2MEN1
SCHEMBL1325515 0.84 MEN1 (0.43) AKR1C3AKR1C2ALDH1A1SMN1; SMN2MEN1
SCHEMBL17186108 0.81 HTT (0.49) ALOX15HTTALDH1A1PABPC1PLK1
SCHEMBL6041219 0.78 MEN1 (0.40) AKR1C3AKR1C2ALDH1A1SMN1; SMN2MEN1
SCHEMBL9382586 0.77 SMN1; SMN2 (0.41) ALDH1A1SMN1; SMN2LMNACYP3A4MEN1
SCHEMBL642839 0.77 SMN1; SMN2 (0.41) ALDH1A1SMN1; SMN2LMNACYP3A4MEN1
SCHEMBL7156656 0.77 HTT (0.39) HTTALDH1A1LMNACYP3A4MEN1
SCHEMBL31048871 0.77 HTT (0.39) HTTALDH1A1LMNACYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0788360-A4 BORONIC ESTER AND ACID COMPOUNDS, SYNTHESIS AND USES PROSCRIPT INC (US) 1998-05-06 EP disclosed
EP-0788360-A1 BORONIC ESTER AND ACID COMPOUNDS, SYNTHESIS AND USES PROSCRIPT, INC. (US) 1997-08-13 EP disclosed