SCHEMBL8709377

SCHEMBL8709377

CCOC(CN(Cc1cccc(OC)c1)S(=O)(=O)c1ccc(C)cc1)OCC

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAS2R14 Q9NYV8 7/20 0.56
CNR2 P34972 2/20 0.50
CA12 O43570 2/20 0.48
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
CA4 P22748 2/20 0.48
CA9 Q16790 2/20 0.48
ALDH1A1 P00352 3/20 0.47
POLB P06746 2/20 0.47
GAA P10253 1/20 0.47
CXCR3 P49682 1/20 0.46
MAPT P10636 1/20 0.45
PKM P14618 1/20 0.45
PTGER1 P34995 1/20 0.45
LMNA P02545 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6769019 0.90 TAS2R14 (0.58) TAS2R14CNR2CA12CA1CA2
SCHEMBL17030819 0.85 CNR2 (0.64) TAS2R14CNR2POLB
SCHEMBL11722886 0.82 CNR2 (0.55) TAS2R14CNR2CA12CA1CA2
SCHEMBL9623455 0.79 CNR2 (0.53) TAS2R14CNR2CA12CA1CA2
SCHEMBL16636846 0.77 CNR2 (0.51) CNR2CA12CA1CA2CA4
SCHEMBL22451561 0.77 TAS2R14 (0.64) TAS2R14CNR2CA12CA1CA2
SCHEMBL6121647 0.76 TAS2R14 (0.79) TAS2R14CNR2CA12CA1CA2
SCHEMBL11497159 0.75 CNR2 (0.63) TAS2R14CNR2ALDH1A1POLBMAPT
SCHEMBL20379430 0.74 LMNA (0.47) TAS2R14CNR2ALDH1A1POLBCXCR3
SCHEMBL12205672 0.73 CNR2 (0.56) TAS2R14CNR2POLBMAPTPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0646119-B1 QUATERNARY NITROGEN-CONTAINING PHOSPHONATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM AS WELL AS DENTAL CALCULUS AND PLAQUE PROCTER & GAMBLE PHARMA (US) 1998-07-15 EP disclosed
EP-0849272-A1 Quaternary nitrogen-containing phosphonate compounds for treating abnormal calcium and phosphate metabolism as well as dental calculus and plaque Procter & Gamble Pharmaceuticals, Inc. (US) 1998-06-24 EP disclosed
US-5770586-A Quaternary nitrogen-containing phosphonate compounds, pharmaceutical compositions, and methods of treating abnormal calcium and phosphate metabolism amd methods of treating and preventing dental calculus and plaque THE PROCTER & GAMBLE COMPANY (US) 1998-06-23 US disclosed
US-5763611-A TREATING OSTEOPOROSIS, RHEUMATOID ARTHRITIS THE PROCTER & GAMBLE COMPANY (US) 1998-06-09 US disclosed
EP-0646119-A1 QUATERNARY NITROGEN-CONTAINING PHOSPHONATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM AS WELL AS DENTAL CALCULUS AND PLAQUE PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1995-04-05 EP disclosed
EP-0642520-A1 THIO-SUBSTITUTED CYCLIC PHOSPHONATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM PROCTER & GAMBLE PHARMACEUTICALS (US) 1995-03-15 EP disclosed
US-5391743-A Treating osteoporosis, rheumatoid arthritis, osteoarthritis PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1995-02-21 US disclosed
WO-1993024498-A1 QUATERNARY NITROGEN-CONTAINING PHOSPHONATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM AS WELL AS DENTAL CALCULUS AND PLAQUE PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1993-12-09 WO disclosed
WO-1993024497-A1 THIO-SUBSTITUTED CYCLIC PHOSPHONATE COMPOUNDS FOR TREATING ABNORMAL CALCIUM AND PHOSPHATE METABOLISM PROCTER & GAMBLE PHARMACEUTICALS, INC. (US) 1993-12-09 WO disclosed