SCHEMBL8709649

SCHEMBL8709649

C/C(=N\O)N(C(=O)[C@H](C)N)[C@@H](CCCCN)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GSR P00390 1/20 0.40
CPB2 Q96IY4 5/20 0.38
RNPEP Q9H4A4 1/20 0.36
FOLH1 Q04609 1/20 0.33
LTA4H P09960 1/20 0.33
GABRR1 P24046 2/20 0.32
NOS2 P35228 4/20 0.31
NOS1 P29475 3/20 0.31
NOS3 P29474 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
TSHR P16473 1/20 0.31
BLM P54132 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716233 0.82 RNPEP (0.40) GSRCPB2RNPEPFOLH1GABRR1
SCHEMBL7224443 0.81 CPB2 (0.41) GSRCPB2RNPEPFOLH1NOS2
SCHEMBL7226730 0.81 CPB2 (0.38) GSRCPB2RNPEPFOLH1
SCHEMBL28210616 0.80 GSR (0.42) GSRCPB2RNPEPFOLH1LTA4H
D-Alanine SCHEMBL4086747 0.79 GSR (0.47) GSRCPB2RNPEPFOLH1LTA4H
Alanine SCHEMBL28591585 0.79 GSR (0.47) GSRCPB2RNPEPFOLH1LTA4H
SCHEMBL8712693 0.78 CPB2 (0.37) GSRCPB2RNPEPFOLH1GABRR1
SCHEMBL8714819 0.78 CPB2 (0.43) GSRCPB2RNPEPFOLH1GABRR1
SCHEMBL28497209 0.76 GSR (0.47) GSRCPB2RNPEPFOLH1LTA4H
SCHEMBL16862530 0.76 GSR (0.38) GSRCPB2RNPEPLTA4HGABRR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885188-A1 HYDROXYAMIDINO DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1998-12-23 EP disclosed
WO-1997032844-A1 HYDROXYAMIDINO DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1997-09-12 WO disclosed