SCHEMBL8714819

SCHEMBL8714819

C/C(=N\O)N(O)[C@@H](CCCCN)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CPB2 Q96IY4 5/20 0.43
GSR P00390 1/20 0.42
RNPEP Q9H4A4 1/20 0.41
FOLH1 Q04609 1/20 0.36
GABRR1 P24046 2/20 0.32
PAOX Q6QHF9 1/20 0.32
SLC6A5 Q9Y345 1/20 0.32
NOS2 P35228 3/20 0.32
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
BLM P54132 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL468723 0.83 CPB2 (0.47) CPB2GSRRNPEPFOLH1GABRR1
SCHEMBL468721 0.83 CPB2 (0.47) CPB2GSRRNPEPFOLH1GABRR1
SCHEMBL8707562 0.80 CPB2 (0.45) CPB2GSRRNPEPFOLH1GABRR1
SCHEMBL8821909 0.80 CPB2 (0.38) CPB2GSRRNPEPFOLH1
SCHEMBL8708989 0.80 CPB2 (0.38) CPB2GSRRNPEPNOS2NOS3
SCHEMBL8716233 0.79 RNPEP (0.40) CPB2GSRRNPEPFOLH1GABRR1
SCHEMBL8709649 0.78 GSR (0.40) CPB2GSRRNPEPFOLH1GABRR1
SCHEMBL7226730 0.78 CPB2 (0.38) CPB2GSRRNPEPFOLH1SLC6A5
SCHEMBL7224443 0.78 CPB2 (0.41) CPB2GSRRNPEPFOLH1NOS2
SCHEMBL7218411 0.78 CPB2 (0.36) CPB2GSRRNPEPFOLH1PAOX

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885188-A1 HYDROXYAMIDINO DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1998-12-23 EP disclosed
WO-1997032844-A9 HYDROXYAMIDINO DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS 1997-12-24 WO disclosed
WO-1997032844-A1 HYDROXYAMIDINO DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1997-09-12 WO disclosed