SCHEMBL8716233

SCHEMBL8716233

C/C(=N\O)N(C(=O)CCCN)[C@@H](CCCCN)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RNPEP Q9H4A4 1/20 0.40
CPB2 Q96IY4 5/20 0.39
GSR P00390 1/20 0.38
FOLH1 Q04609 1/20 0.36
PAOX Q6QHF9 1/20 0.33
SLC6A5 Q9Y345 1/20 0.32
CYP1A2 P05177 2/20 0.32
LMNA P02545 2/20 0.32
THRB P10828 2/20 0.32
BLM P54132 2/20 0.32
KMT2A Q03164 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
GABRR3 A8MPY1 1/20 0.32
GABRP O00591 1/20 0.32
GABRD O14764 1/20 0.32
HDAC3 O15379 1/20 0.32
GABBR2 O75899 1/20 0.32
GABRA1 P14867 1/20 0.32
TSHR P16473 1/20 0.32
GABRB1 P18505 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709649 0.82 GSR (0.40) RNPEPCPB2GSRFOLH1CYP1A2
SCHEMBL7226730 0.82 CPB2 (0.38) RNPEPCPB2GSRFOLH1SLC6A5
SCHEMBL7224443 0.82 CPB2 (0.41) RNPEPCPB2GSRFOLH1
SCHEMBL8712693 0.80 CPB2 (0.37) RNPEPCPB2GSRFOLH1GABRR1
SCHEMBL8714819 0.79 CPB2 (0.43) RNPEPCPB2GSRFOLH1PAOX
SCHEMBL8931801 0.78 SLC6A5 (0.45) RNPEPCPB2GSRSLC6A5
SCHEMBL8931799 0.78 SLC6A5 (0.45) RNPEPCPB2GSRSLC6A5
SCHEMBL1886103 0.77 GSR (0.43) RNPEPCPB2GSRFOLH1SLC6A5
SCHEMBL1886100 0.77 GSR (0.43) RNPEPCPB2GSRFOLH1SLC6A5
SCHEMBL9314956 0.77 SLC6A5 (0.47) CPB2GSRSLC6A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0885188-A1 HYDROXYAMIDINO DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1998-12-23 EP disclosed
WO-1997032844-A1 HYDROXYAMIDINO DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1997-09-12 WO disclosed