SCHEMBL8710247

SCHEMBL8710247

C[Si](C)(C)CCOCOc1cccnc1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR4 O95977 1/20 0.44
KDM4E B2RXH2 5/20 0.35
LMNA P02545 5/20 0.35
MAPT P10636 6/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 4/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
RAB9A P51151 4/20 0.33
NPC1 O15118 3/20 0.33
HTT P42858 2/20 0.32
TRIM24 O15164 1/20 0.32
TRIM33 Q9UPN9 1/20 0.32
KDM1A O60341 1/20 0.31
DGAT1 O75907 1/20 0.31
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31437246 1.00 S1PR4 (0.44) S1PR4KDM4ELMNAMAPTCYP1A2
SCHEMBL4858597 0.85 S1PR4 (0.43) S1PR4KDM4ELMNAMAPTCYP1A2
SCHEMBL34475296 0.81 HTR7 (0.47) KDM4ELMNAMAPTCYP1A2CYP3A4
SCHEMBL24538043 0.81 HTR7 (0.47) KDM4ELMNAMAPTCYP1A2CYP3A4
SCHEMBL570791 0.80 S1PR4 (0.45) S1PR4KDM4ELMNAMAPTCYP1A2
SCHEMBL25236185 0.79 KDM4E (0.43) KDM4ELMNAMAPTCYP1A2CYP3A4
SCHEMBL31022737 0.79 KDM4E (0.43) KDM4ELMNAMAPTCYP1A2CYP3A4
SCHEMBL30557100 0.78 KDM4E (0.35) KDM4ELMNAMAPTCYP1A2CYP3A4
SCHEMBL26118784 0.78 KDM4E (0.35) KDM4ELMNAMAPTCYP1A2CYP3A4
SCHEMBL9476261 0.78 PLCG1 (0.35) MAPTSMN1; SMN2ALOX5APFEN1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250304537-A1 HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME REPARE THERAPEUTICS INC. (CA) 2025-10-02 US disclosed
EP-4526293-A1 HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME Repare Therapeutics Inc. (CA) 2025-03-26 EP disclosed
WO-2023220831-A1 HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME REPARE THERAPEUTICS INC. (CA) 2023-11-23 WO disclosed
US-20230174536-A1 NOVEL COMPOUNDS FOR DIAGNOSIS AC IMMUNE SA (CH) 2023-06-08 US disclosed
EP-1516874-B1 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation DOW AGROSCIENCES LLC (US) 2015-08-19 EP disclosed
US-RE39991-E1 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation DOW AGROSCIENCES LLC (US) 2008-01-01 US disclosed
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250304537-A1 HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME CSNK1A1, CSNK1G1, CSNK2A1 S1PR4 4126/4885KDM4E 2698/4885LMNA 3295/4885
US-20230174536-A1 NOVEL COMPOUNDS FOR DIAGNOSIS SNCA, PARK7, SLC6A3 S1PR4 1346/4885KDM4E 4851/4885LMNA 1661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.