SCHEMBL8710852

SCHEMBL8710852

O=C(c1ccc(F)cc1)C1CCN(CCN(C(=O)c2ccc([N+](=O)[O-])cc2)c2cccnc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.51
HTR2A P28223 4/20 0.51
SLC18A3 Q16572 3/20 0.47
ACHE P22303 1/20 0.47
HTR2C P28335 2/20 0.45
HTR7 P34969 1/20 0.45
HTR6 P50406 1/20 0.45
KDM4E B2RXH2 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8711151 0.93 HTR2A (0.57) HSD11B1HTR2ASLC18A3ACHE
SCHEMBL8715718 0.89 HTR2A (0.61) HSD11B1HTR2AACHEKDM4ECYP1A2
SCHEMBL9232680 0.89 HSD11B1 (0.56) HSD11B1HTR2AACHEHTR2CHTR7
SCHEMBL8712117 0.88 HSD11B1 (0.59) HSD11B1HTR2AACHEHTR2CHTR7
SCHEMBL8710951 0.88 SLC18A3 (0.50) HTR2ASLC18A3ACHEHTR2CHTR7
SCHEMBL8711319 0.87 SLC18A3 (0.49) HSD11B1HTR2ASLC18A3HTR2CHTR7
SCHEMBL8710844 0.85 SLC18A3 (0.48) HTR2ASLC18A3HTR2CHTR7HTR6
SCHEMBL8711236 0.85 SLC18A3 (0.47) HTR2ASLC18A3HTR2CHTR7HTR6
SCHEMBL8713817 0.85 MEN1 (0.49) HTR2ASLC18A3HTR2CHTR7HTR6
SCHEMBL8714509 0.85 HSD11B1 (0.51) HSD11B1HTR2AACHEHTR2CHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed