SCHEMBL8710952

SCHEMBL8710952

COc1ccc(S(=O)(=O)N(CCO)c2ccccc2OC)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.60
ALDH1A1 P00352 3/20 0.55
LMNA P02545 2/20 0.55
HPGD P15428 2/20 0.55
HTT P42858 1/20 0.55
SMN1; SMN2 Q16637 2/20 0.54
MAPT P10636 2/20 0.54
MEN1 O00255 1/20 0.54
KMT2A Q03164 1/20 0.54
KEAP1 Q14145 7/20 0.54
NFE2L2 Q16236 7/20 0.54
GAA P10253 2/20 0.51
NPSR1 Q6W5P4 2/20 0.51
USP2 O75604 1/20 0.51
TSHR P16473 1/20 0.51
MMP1 P03956 1/20 0.50
MMP7 P09237 1/20 0.50
MMP8 P22894 1/20 0.50
MMP12 P39900 1/20 0.50
MMP13 P45452 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712282 0.89 ESR1 (0.60) ESR1LMNAHPGDSMN1; SMN2KMT2A
SCHEMBL1629150 0.83 KEAP1 (0.77) KEAP1NFE2L2
SCHEMBL10300192 0.79 ESR1 (0.49) ESR1ALDH1A1LMNAHPGDSMN1; SMN2
SCHEMBL15833703 0.79 SMN1; SMN2 (0.65) ALDH1A1LMNASMN1; SMN2MAPTKEAP1
SCHEMBL8714947 0.78 ESR1 (0.63) ESR1ALDH1A1LMNAHPGDHTT
SCHEMBL6096889 0.78 SMN1; SMN2 (0.54) ALDH1A1HPGDHTTSMN1; SMN2MEN1
SCHEMBL6096893 0.78 SMN1; SMN2 (0.54) ALDH1A1HPGDHTTSMN1; SMN2MEN1
SCHEMBL6096525 0.77 MET (0.69) SMN1; SMN2KEAP1NFE2L2NPSR1MMP1
SCHEMBL6096531 0.77 MET (0.69) SMN1; SMN2KEAP1NFE2L2NPSR1MMP1
SCHEMBL4936946 0.76 SMN1; SMN2 (0.77) LMNAHTTSMN1; SMN2KEAP1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed