SCHEMBL8714947

SCHEMBL8714947

COc1ccccc1N(CO)S(=O)(=O)c1ccc(F)cc1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.63
KEAP1 Q14145 1/20 0.52
NFE2L2 Q16236 1/20 0.52
KMT2A Q03164 3/20 0.51
TSHR P16473 2/20 0.51
MAPK1 P28482 1/20 0.51
HSD17B10 Q99714 1/20 0.51
MAPT P10636 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
MEN1 O00255 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
CRHBP P24387 1/20 0.49
CRHR2 Q13324 1/20 0.49
ALDH1A1 P00352 3/20 0.49
HPGD P15428 2/20 0.49
HTT P42858 2/20 0.49
LMNA P02545 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712282 0.89 ESR1 (0.60) ESR1KEAP1NFE2L2KMT2ATSHR
SCHEMBL18101489 0.81 SMN1; SMN2 (0.70) TSHRMAPTSMN1; SMN2ALDH1A1HPGD
SCHEMBL8710952 0.78 ESR1 (0.60) ESR1KEAP1NFE2L2KMT2ATSHR
SCHEMBL1629150 0.77 KEAP1 (0.77) KEAP1NFE2L2
SCHEMBL2174816 0.76 SMN1; SMN2 (0.57) KMT2AMAPTSMN1; SMN2MEN1ALDH1A1
SCHEMBL9226646 0.72 HTR7 (0.59)
SCHEMBL16557468 0.72 HPGD (0.81) TSHRMAPTSMN1; SMN2ALDH1A1HPGD
SCHEMBL1040894 0.71 HCRTR2 (0.62) ESR1KEAP1NFE2L2KMT2AMEN1
SCHEMBL14470046 0.70 KMT2A (0.56) KEAP1NFE2L2KMT2ATSHRMAPK1
SCHEMBL6801637 0.70 NR3C1 (0.63) KEAP1NFE2L2KMT2AMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed